SCHEMBL1026533

SCHEMBL1026533

CC(=O)N(Cc1cccc(N)c1)Cc1cccc(N(C(=O)OC(=O)C(F)(F)F)C(C)(C)C)c1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
HDAC6 Q9UBN7 1/20 0.31
CETP P11597 1/20 0.31
MGLL Q99685 1/20 0.31
KMT2A Q03164 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL1026532 0.84 CRHBP (0.40) HSD11B1CRHBPCRHR2KMT2AL3MBTL1
SCHEMBL1023948 0.80 CTSC (0.35)
SCHEMBL1026531 0.77 ALDH1A1 (0.41) HSD11B1HDAC6MGLLL3MBTL1
SCHEMBL1028316 0.70 OPRM1 (0.43) KMT2A
SCHEMBL1026191 0.69 MAOA (0.50) HSD11B1CRHBPCRHR2KMT2AL3MBTL1
Trifluoroacetic Acid SCHEMBL1026530 0.69 ALDH1A1 (0.44) HDAC6L3MBTL1
SCHEMBL1026880 0.69 THRA (0.39) HSD11B1CRHBPCRHR2KMT2AL3MBTL1
SCHEMBL13623194 0.67 AURKA (0.44) HDAC6
SCHEMBL1026509 0.66 CYP1A2 (0.36) HSD11B1CRHBPCRHR2KMT2AL3MBTL1
SCHEMBL6956921 0.66 GRIN2D (0.45) HSD11B1HDAC6KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274288-A2 MACROCYCLIC COMPOUNDS AND THEIR USE AS KINASE INHIBITORS Incyte Corporation (US) 2011-01-19 EP disclosed