SCHEMBL10242251

SCHEMBL10242251

CN1C(=O)NCC1c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 9/20 0.42
ATM Q13315 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
KCNH2 Q12809 2/20 0.37
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
RECQL P46063 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19694652 0.85 HTR2C (0.46) ATMNPSR1RECQL
SCHEMBL15743974 0.74 TACR1 (0.40) TACR1KCNH2
SCHEMBL13394555 0.74 TACR1 (0.33) TACR1ATMNPSR1KCNH2
SCHEMBL6958220 0.71 P2RX7 (0.40)
SCHEMBL20956906 0.70 ABCC9 (0.43)
SCHEMBL2385210 0.70 TACR1 (0.47) TACR1
SCHEMBL20780480 0.70 TACR1 (0.37) TACR1KCNH2
SCHEMBL13413567 0.70 TACR1 (0.37) TACR1
SCHEMBL7018969 0.68 CYP19A1 (0.44)
SCHEMBL20794021 0.68 ADRB1 (0.37) TACR1KCNH2RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765793-B1 ANACETRAPIB AND OTHER CETP INHIBITPRS MERCK SHARP & DOHME (US) 2012-09-26 EP disclosed
EP-2415759-A1 CETP inhibitors Merck Sharp & Dohme Corporation (US) 2012-02-08 EP disclosed