SCHEMBL7018969

SCHEMBL7018969

CN1C(=O)NCC1c1ccc(N)cc1

nearest known ligand 0.44

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 7/20 0.44
DDB1 Q16531 1/20 0.37
CRBN Q96SW2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5309109 0.83 CYP19A1 (0.41) CYP19A1DDB1CRBN
SCHEMBL7058755 0.80 DDB1 (0.42) DDB1CRBN
Hydrochloric Acid SCHEMBL31029179 0.77 CYP19A1 (0.40) CYP19A1DDB1CRBN
SCHEMBL6958220 0.75 P2RX7 (0.40)
SCHEMBL6619946 0.73 PTGS2 (0.41)
SCHEMBL30912484 0.71 KDM4E (0.54) CYP19A1DDB1CRBN
SCHEMBL30912593 0.71 KDM4E (0.54) CYP19A1DDB1CRBN
SCHEMBL30912576 0.71 KDM4E (0.54) CYP19A1DDB1CRBN
SCHEMBL26548245 0.69 CYP19A1 (0.45) CYP19A1
SCHEMBL19694652 0.67 HTR2C (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3066098-A1 SUBSTITUTED URACILS AND USE THEREOF Bayer Pharma Aktiengesellschaft (DE) 2016-09-14 EP disclosed
WO-2015067630-A1 SUBSTITUTED URACILS AND USE THEREOF BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-05-14 WO disclosed
EP-1326865-A2 AZA- AND POLYAZA-NAPHTHALENYL CARBOXAMIDES USEFUL AS HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2003-07-16 EP disclosed
WO-2002030930-A2 AZA- AND POLYAZA-NAPHTHALENYL CARBOXAMIDES USEFUL AS HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 2002-04-18 WO disclosed