SCHEMBL10242437

SCHEMBL10242437

Cc1cc(-c2ccc3ncc(C(C)(F)c4ccc5ncccc5c4)n3n2)on1

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MET P08581 20/20 0.55
NQO2 P16083 1/20 0.44
PDE3B Q13370 1/20 0.44
PDE3A Q14432 1/20 0.44
PIP4K2C Q8TBX8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2697690 0.93 MET (0.55) METNQO2PDE3BPDE3APIP4K2C
SCHEMBL10242494 0.85 MET (0.58) METNQO2PDE3BPDE3APIP4K2C
SCHEMBL2698486 0.81 MET (0.68) METNQO2PDE3BPDE3APIP4K2C
SCHEMBL2697816 0.77 MET (0.64) MET
SCHEMBL2698979 0.75 TGFBR1 (0.42) MET
SCHEMBL10242535 0.75 MET (0.59) METNQO2PDE3BPDE3APIP4K2C
SCHEMBL10242426 0.75 MET (0.81) METNQO2PDE3BPDE3APIP4K2C
SCHEMBL2697147 0.71 MET (1.00) METNQO2PDE3BPDE3APIP4K2C
SCHEMBL1658513 0.71 MET (0.78) METNQO2PDE3BPDE3APIP4K2C
SCHEMBL3411435 0.70 MET (0.53) METNQO2PDE3BPDE3APIP4K2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120107275-A1 FUSED HETEROCYCLIC DERIVATIVES AND METHODS OF USE AMGEN INC. (US) 2012-05-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120107275-A1 FUSED HETEROCYCLIC DERIVATIVES AND METHODS OF USE HGF, HGFAC, MET MET 3/4885NQO2 1016/4885PDE3B 1730/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.