SCHEMBL10242614

SCHEMBL10242614

Fc1c(Br)ccc2c1NCC2

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.38
HTR2C P28335 5/20 0.38
HTR2B P41595 4/20 0.38
PARP10 Q53GL7 7/20 0.37
PARP1 P09874 5/20 0.37
PARP11 Q9NR21 2/20 0.33
PNMT P11086 2/20 0.32
ASIC3 Q9UHC3 1/20 0.32
KDM1A O60341 2/20 0.32
KCNH2 Q12809 2/20 0.32
KDM1B Q8NB78 2/20 0.32
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
F7 P08709 1/20 0.30
F3 P13726 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20865736 0.76 ALDH1A1 (0.38) HTR2AHTR2CHTR2BPARP10PARP1
SCHEMBL30664964 0.76 HTR2A (0.38) HTR2AHTR2CHTR2BPARP10PARP1
SCHEMBL7657136 0.76 HTR2A (0.38) HTR2AHTR2CHTR2BPARP10PARP1
SCHEMBL652655 0.71 PARP10 (0.43) HTR2AHTR2CHTR2BPARP10PARP1
SCHEMBL31393728 0.69 PARP10 (0.42) HTR2AHTR2CHTR2BPARP10PARP11
SCHEMBL22993473 0.69 PNMT (0.54) HTR2AHTR2CHTR2BPNMTASIC3
SCHEMBL29407560 0.69 PNMT (0.54) HTR2AHTR2CHTR2BPNMTASIC3
SCHEMBL13035941 0.68 FABP6 (0.41) ALDH1A1MAPT
Hydrochloric Acid SCHEMBL23727152 0.68 PNMT (0.53) HTR2AHTR2CHTR2BPNMTASIC3
SCHEMBL23384836 0.68 NOTUM (0.46) HTR2AHTR2CHTR2BPARP10PARP11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260015351-A1 METHODS AND COMPOUNDS FOR INHIBITING MKK7 ENZYMES AXONIS THERAPEUTICS INC (US) 2026-01-15 US disclosed
WO-2024006379-A1 METHODS AND COMPOUNDS FOR INHIBITING MKK7 ENZYMES AXONIS THERAPEUTICS, INC. (US) 2024-01-04 WO disclosed
US-8114846-B2 Combined treatment with an EGFR kinase inhibitor and an agent that sensitizes tumor cells to the effects of EGFR kinase inhibitors OSI Pharmaceuticals, LLC (US) 2012-02-14 US disclosed
US-20100166776-A1 COMBINED TREATMENT WITH AN EGFR KINASE INHIBITOR AND AN AGENT THAT SENSITIZES TUMOR CELLS TO THE EFFECTS OF EGFR KINASE INHIBITORS OSI PHARMACEUTICALS, INC. 2010-07-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100166776-A1 COMBINED TREATMENT WITH AN EGFR KINASE INHIBITOR AND AN AGENT THAT SENSITIZES TUMOR CELLS TO THE EFFECTS OF EGFR KINASE INHIBITORS EGFR, ERBB2, RICTOR HTR2A 3636/4885HTR2C 3925/4885HTR2B 4282/4885
US-20260015351-A1 METHODS AND COMPOUNDS FOR INHIBITING MKK7 ENZYMES PRKCSH, MAPK7, PRKCB HTR2A 4581/4885HTR2C 3132/4885HTR2B 3935/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.