SCHEMBL10243525

SCHEMBL10243525

CCN(CCNC(=O)OC)C(C)c1ccc(OCc2ccccc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.54
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
BCHE P06276 1/20 0.47
L3MBTL1 Q9Y468 2/20 0.46
ACACB O00763 1/20 0.45
MAPT P10636 1/20 0.45
NOX1 Q9Y5S8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10243580 0.86 ACACB (0.49) NPC1RAB9ASMN1; SMN2ACACB
SCHEMBL10243497 0.86 SLC22A1 (0.43) ALOX5SMN1; SMN2
SCHEMBL10244300 0.85 MTNR1A (0.48) NPC1RAB9ASMN1; SMN2
SCHEMBL10244037 0.84 CYP1A2 (0.46) ALOX5NPC1RAB9ASMN1; SMN2
SCHEMBL10244298 0.83 TDP1 (0.42) NPC1RAB9ASMN1; SMN2L3MBTL1MAPT
SCHEMBL10244480 0.81 CYP1A2 (0.43) RAB9ASMN1; SMN2ACACB
SCHEMBL10244079 0.81 ALDH1A1 (0.40) SMN1; SMN2L3MBTL1MAPT
SCHEMBL10243510 0.80 ALOX5 (0.40) ALOX5SMN1; SMN2L3MBTL1
SCHEMBL10243697 0.80 ALDH1A1 (0.43) MAPT
SCHEMBL10243433 0.79 MAPT (0.43) SMN1; SMN2L3MBTL1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8097708-B2 10a-Azalide compound TAISHO PHARMACEUTICAL CO., LTD. (JP) 2012-01-17 US disclosed
US-8097708-B2 10a-Azalide compound TAISHO PHARMACEUTICAL CO., LTD. (JP) 2012-01-17 US disclosed
US-20090281292-A1 10a-Azalide Compound MEIJI SEIKA PHARMA CO., LTD. (JP) 2009-11-12 US disclosed
US-20090281292-A1 10a-Azalide Compound MEIJI SEIKA PHARMA CO., LTD. (JP) 2009-11-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090281292-A1 10a-Azalide Compound IL17A, AZI2, HDAC9 ALOX5 2387/4885NPC1 209/4885RAB9A 5/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.