SCHEMBL10244925

SCHEMBL10244925

Nc1cc(CO)ccc1Oc1cccnc1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.49
ALDH1A1 P00352 2/20 0.49
TTR P02766 1/20 0.48
LMNA P02545 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
PPARD Q03181 1/20 0.45
MKNK1 Q9BUB5 1/20 0.43
MKNK2 Q9HBH9 1/20 0.43
CYP19A1 P11511 4/20 0.42
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTT P42858 1/20 0.38
BRD4 O60885 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8105420 0.82 TTR (0.70) SMN1; SMN2ALDH1A1TTRCYP1A2CYP3A4
SCHEMBL875806 0.80 ALDH1A1 (0.68) SMN1; SMN2ALDH1A1TTRLMNATDP1
SCHEMBL7995147 0.80 SMN1; SMN2 (0.46) SMN1; SMN2ALDH1A1TTRLMNATDP1
SCHEMBL2031421 0.78 ALDH1A1 (0.53) SMN1; SMN2ALDH1A1LMNATDP1CYP19A1
SCHEMBL7390045 0.78 CYP1A2 (0.66) SMN1; SMN2ALDH1A1LMNATDP1CYP19A1
SCHEMBL4938372 0.77 LMNA (0.68) SMN1; SMN2ALDH1A1LMNATDP1MKNK1
SCHEMBL2646628 0.76 ALDH1A1 (0.62) SMN1; SMN2ALDH1A1LMNATDP1CYP19A1
SCHEMBL11478665 0.75 LMNA (0.53) SMN1; SMN2ALDH1A1LMNATDP1CYP19A1
SCHEMBL15779486 0.75 LMNA (0.53) SMN1; SMN2ALDH1A1LMNATDP1CYP19A1
SCHEMBL2933241 0.74 L3MBTL1 (0.60) SMN1; SMN2ALDH1A1LMNATDP1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037782-A1 TRICYCLIC COMPOUNDS, PREPARATION METHODS, AND THEIR USES GLAXO GROUP LIMITED (GB) 2012-03-29 WO disclosed