SCHEMBL7995147

SCHEMBL7995147

OCc1ccc(Oc2cccnc2)c(C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.46
ALDH1A1 P00352 1/20 0.46
PPARD Q03181 1/20 0.45
TTR P02766 1/20 0.44
SUCNR1 Q9BXA5 1/20 0.44
LMNA P02545 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
AR P10275 1/20 0.42
MKNK1 Q9BUB5 1/20 0.40
MKNK2 Q9HBH9 1/20 0.40
CYP19A1 P11511 3/20 0.39
NR1H2 P55055 4/20 0.39
NR1H3 Q13133 4/20 0.39
IDH2 P48735 1/20 0.38
CYP1A2 P05177 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38
S1PR1 P21453 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3900976 0.83 TTR (0.64) TTRARNR1H2NR1H3
SCHEMBL10244925 0.80 SMN1; SMN2 (0.49) SMN1; SMN2ALDH1A1PPARDTTRLMNA
SCHEMBL14021961 0.80 SMN1; SMN2 (0.49) SMN1; SMN2ALDH1A1PPARDSUCNR1LMNA
SCHEMBL8004583 0.79 AOC3 (0.49) SMN1; SMN2SUCNR1
SCHEMBL883499 0.78 EPAS1 (0.49) SMN1; SMN2ALDH1A1TTRARNR1H2
Hydrochloric Acid SCHEMBL8104657 0.78 AOC3 (0.50) SMN1; SMN2SUCNR1
SCHEMBL9889486 0.77 AR (0.48) ALDH1A1TTRARNR1H2NR1H3
SCHEMBL8004575 0.77 SMN1; SMN2 (0.45) SMN1; SMN2PPARDSUCNR1IDH2CYP1A2
SCHEMBL875806 0.76 ALDH1A1 (0.68) SMN1; SMN2ALDH1A1PPARDTTRLMNA
Hydrochloric Acid SCHEMBL8097516 0.76 SMN1; SMN2 (0.45) SMN1; SMN2PPARDSUCNR1IDH2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0748795-B1 Substituted benzyloxycarbonyl guanidines as Na+/H+ exchange inhibitors, process for their preparation, their use as medicinal or diagnostic agents as well as medicament containing them HOECHST AG (DE) 2000-08-23 EP disclosed
US-6022899-A EFFECTIVE INHIBITORS OF THE CELLULAR SODIUM PROTON ANTIPORTER HOECHST AKTIENGESELLSCHAFT (DE) 2000-02-08 US disclosed
US-5753710-A INHIBITORS OF THE CELLULAR SODIUM PROTON ANTIPORTER HOECHST AKTIENGESELLSCHAFT (DE) 1998-05-19 US disclosed
EP-0748795-A2 Substituted benzyloxycarbonyl guanidines as Na+/H+ exchange inhibitors, process for their preparation, their use as medicinal or diagnostic agents as well as medicament containing them HOECHST AKTIENGESELLSCHAFT (DE) 1996-12-18 EP disclosed