SCHEMBL10247611

SCHEMBL10247611

C=Cc1ccc(-c2ccc(C(N)=O)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA9 Q16790 1/20 0.50
CA14 Q9ULX7 1/20 0.50
ERN1 O75460 2/20 0.47
MKNK1 Q9BUB5 7/20 0.47
MKNK2 Q9HBH9 7/20 0.47
PARP10 Q53GL7 2/20 0.47
PARP3 Q9Y6F1 1/20 0.47
ALDH1A1 P00352 2/20 0.46
CYP17A1 P05093 1/20 0.44
HDAC2 Q92769 1/20 0.44
BRD4 O60885 1/20 0.44
BRD9 Q9H8M2 1/20 0.44
KMT2A Q03164 1/20 0.43
PARP15 Q460N3 1/20 0.43
PARP14 Q460N5 1/20 0.43
PARP16 Q8N5Y8 1/20 0.43
PARP11 Q9NR21 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10243239 1.00 CA12 (0.50) CA12CA1CA2CA9CA14
SCHEMBL1051273 0.94 ALDH1A1 (0.52) CA1CA2PARP10PARP3ALDH1A1
SCHEMBL30053335 0.91 PARP10 (0.50) CA1CA2PARP10PARP3ALDH1A1
Trimethylammonium SCHEMBL461393 0.86 PARP10 (0.46) CA1CA2PARP10PARP3ALDH1A1
Terephthalamide SCHEMBL28201048 0.83 TSHR (0.60) CA1CA2MKNK1MKNK2PARP10
SCHEMBL15764248 0.82 ERN1 (0.55) ERN1HDAC2PARP1
SCHEMBL1002578 0.82 CA2 (0.67) CA12CA1CA2CA9CA14
SCHEMBL10245562 0.81 ALDH1A1 (0.56) CA12CA1CA2CA9CA14
SCHEMBL19048679 0.81 PARP10 (0.69) CA12CA1CA2CA9CA14
SCHEMBL1676005 0.81 ALDH1A1 (0.56) CA12CA1CA2CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012018868-A1 SUBSTITUTED 2-HYDROXY-4-(2-(PHENYLSULFONAMIDO)ACETAMIDO)BENZOIC ACID ANALOGS AS INHIBITORS OF STAT PROTEINS UNIVERSITY OF CENTRAL FLORIDA RESEARCH FOUNDATION, INC. (US) 2012-02-09 WO disclosed