SCHEMBL10248963

SCHEMBL10248963

CC(C)c1nc(N)n(Cc2ccc(Cl)cc2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.49
GAA P10253 1/20 0.49
GFER P55789 1/20 0.49
SMN1; SMN2 Q16637 4/20 0.43
MAPT P10636 3/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
LMNA P02545 2/20 0.41
STAT3 P40763 1/20 0.41
TNF P01375 1/20 0.40
CXCL8 P10145 1/20 0.40
SOS1 Q07889 1/20 0.40
NOD2 Q9HC29 1/20 0.40
NOD1 Q9Y239 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A3 Q01959 1/20 0.40
TSHR P16473 1/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HSP90AB1 P08238 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10284722 0.79 POLB (0.57) POLBGAAGFERSMN1; SMN2MAPT
SCHEMBL21793295 0.68 KMT2A (0.51) POLBGAASMN1; SMN2MAPTMEN1
SCHEMBL31272007 0.68 MAPT (0.47) POLBGAAGFERSMN1; SMN2MAPT
SCHEMBL31272189 0.67 MET (0.45) SMN1; SMN2MAPTMEN1KMT2A
SCHEMBL31272220 0.67 MAPT (0.43) POLBMAPTMEN1KMT2ALMNA
SCHEMBL8035176 0.66 GAA (0.76) POLBGAAGFERSMN1; SMN2MAPT
SCHEMBL11655968 0.66 GAA (1.00) POLBGAAGFERSMN1; SMN2MAPT
SCHEMBL3169680 0.66 POLB (0.61) POLBGAAGFERSMN1; SMN2MAPT
SCHEMBL1801043 0.66 GAA (0.76) POLBGAAGFERSMN1; SMN2MAPT
SCHEMBL31272068 0.65 NFKB1 (0.41) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8124610-B2 Sodium channel inhibitors ICAGEN INC. (US) 2012-02-28 US disclosed
US-20090023740-A1 SODIUM CHANNEL INHIBITORS ICAGEN (US) 2009-01-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090023740-A1 SODIUM CHANNEL INHIBITORS TRPV1, SCN1A, SCN2A POLB 4439/4885GAA 3730/4885GFER 976/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.