SCHEMBL1025663

SCHEMBL1025663

Cn1nc(N)c(-c2ccc(F)cc2Cl)c1-c1ccc(Cl)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.40
SCN10A Q9Y5Y9 1/20 0.40
HSD11B1 P28845 2/20 0.39
HTT P42858 1/20 0.38
NR1H2 P55055 1/20 0.38
NR1H3 Q13133 1/20 0.38
SRC P12931 2/20 0.38
BRAF P15056 2/20 0.38
KDR P35968 2/20 0.38
GRM5 P41594 2/20 0.37
RIPK2 O43353 1/20 0.37
EGFR P00533 1/20 0.37
TNK2 Q07912 1/20 0.37
PTK6 Q13882 1/20 0.37
MINK1 Q8N4C8 1/20 0.37
CLK1 P49759 1/20 0.37
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
TP53 P04637 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1025414 0.87 HSD11B1 (0.41) HSD11B1NR1H2NR1H3GRM5KDM4E
SCHEMBL19953206 0.73 POLB (0.38) HTT
SCHEMBL173503 0.71 HSD11B1 (0.47) DPP4SCN10AHSD11B1IGF1R
SCHEMBL29520229 0.71 HSD11B1 (0.47) DPP4SCN10AHSD11B1
SCHEMBL173619 0.71 HSD11B1 (0.47) DPP4SCN10AHSD11B1
SCHEMBL20075418 0.71 MAPK14 (0.44) HTTGRM5KDM4ESMN1; SMN2
SCHEMBL8025221 0.71 HTT (0.46) HTTNR1H2NR1H3SRCKDR
SCHEMBL2340641 0.70 GRM5 (0.38) GRM5SMN1; SMN2
SCHEMBL21711491 0.70 SLC34A1 (0.47) DPP4SCN10AHSD11B1GRM5CLK1
SCHEMBL6177712 0.70 MAPK14 (0.65) SRCBRAFKDRRIPK2EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274285-A1 NOVEL PYRAZOLE DERIVATIVES Syngenta Participations AG (CH) 2011-01-19 EP disclosed
WO-2009127612-A1 NOVEL PYRAZOLE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2009-10-22 WO disclosed