SCHEMBL19953206

SCHEMBL19953206

COc1cc(F)c(-c2c(N)nn(C)c2-c2ccc(Cl)cc2)c(F)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.38
HTT P42858 1/20 0.38
CA1 P00915 3/20 0.36
CA2 P00918 3/20 0.36
PTGS1 P23219 2/20 0.36
PTGS2 P35354 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
BACE1 P56817 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36
THPO P40225 1/20 0.36
BLM P54132 1/20 0.36
PMP22 Q01453 1/20 0.36
HIF1A Q16665 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
ADORA1 P30542 1/20 0.36
MAPT P10636 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1023884 0.87 CYP1A2 (0.38) PTGS1PTGS2NPSR1BACE1CYP1A2
SCHEMBL1023575 0.81 L3MBTL1 (0.39) POLBPTGS1PTGS2NPSR1BACE1
SCHEMBL1027586 0.75 GRM8 (0.36) PTGS2BACE1CYP1A2PDE10A
SCHEMBL1024672 0.74 L3MBTL1 (0.39) POLBPTGS1PTGS2NPSR1BACE1
SCHEMBL1025663 0.73 DPP4 (0.40) HTT
SCHEMBL1025606 0.73 GRM5 (0.38) MAPT
SCHEMBL1026639 0.73 PDE10A (0.37) CYP1A2MAPTMEN1KMT2APDE10A
SCHEMBL1023290 0.72 NR1H2 (0.36) PTGS2PDE10A
SCHEMBL13165379 0.70 MEN1 (0.47) CA1CA2NPSR1CYP1A2CYP3A4
SCHEMBL30941226 0.70 THRB (0.41) NPSR1CYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018048969-A1 MULTI-TARGETED HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2018-03-15 WO disclosed