SCHEMBL1025834

SCHEMBL1025834

Nc1cccnc1C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.46
HSD17B10 Q99714 1/20 0.46
KDM4E B2RXH2 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
TLR7 Q9NYK1 1/20 0.38
NOS3 P29474 3/20 0.38
NOS2 P35228 3/20 0.38
POLB P06746 2/20 0.37
NOS1 P29475 2/20 0.37
KMT2A Q03164 4/20 0.36
HSP90AA1 P07900 3/20 0.36
MEN1 O00255 3/20 0.36
MAPT P10636 3/20 0.36
HSP90AB1 P08238 2/20 0.36
LMNA P02545 1/20 0.36
BLM P54132 1/20 0.36
HIF1A Q16665 1/20 0.36
PI4KA P42356 1/20 0.36
PI4K2B Q8TCG2 1/20 0.36
PI4K2A Q9BTU6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20689253 0.83 NOS3 (0.39) HTTHSD17B10KDM4EL3MBTL1TLR7
SCHEMBL28513854 0.81 PDE10A (0.41) HTTHSD17B10KDM4EL3MBTL1KMT2A
SCHEMBL30615592 0.79 HTT (0.39) HTTHSD17B10KDM4EL3MBTL1TLR7
SCHEMBL29581438 0.79 MAPT (0.47) HTTHSD17B10KDM4EL3MBTL1KMT2A
SCHEMBL21463674 0.79 HTT (0.39) HTTHSD17B10KDM4EL3MBTL1TLR7
SCHEMBL5178183 0.78 HTT (0.41) HTTHSD17B10KDM4EL3MBTL1TLR7
SCHEMBL7803270 0.77 NOS3 (0.41) HTTKDM4ENOS3NOS2NOS1
SCHEMBL10515301 0.77 ALDH1A1 (0.39) HTTKDM4ENOS3NOS2NOS1
SCHEMBL30113073 0.77 HTT (0.46) HTTHSD17B10KDM4EL3MBTL1TLR7
SCHEMBL16914429 0.74 PSMD14 (0.45) HTTHSD17B10KDM4EL3MBTL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 155 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025125665-A1 FURTHER SUBSTITUTED IMIDAZOLES AS INHIBITORS OF NAV1.8 Grünenthal GmbH (DE) 2025-06-19 WO claimed
CN-102977009-B A kind of synthetic method of 2-trifluoromethyl-3-fluorine pyridine Ao Sainuo bio tech ltd, Hangzhou (CN) 2015-07-29 CN claimed
CN-102977009-A Synthesizing method of 2-trifluoromethyl-3-fluoropyridin HANGZHOU ALLSINO CHEMICAL CO LTD 2013-03-20 CN claimed
EP-1252889-B1 REMEDIES OR PREVENTIVES FOR PULMONARY INSUFFICIENCY CONTAINING DIAMINOTRIFLUOROMETHYLPYRIDINE DERIVATIVES ISHIHARA SANGYO KAISHA (JP) 2006-08-09 EP claimed
US-20030109551-A1 Remedies or preventives for pulmonary insufficiency containing diaminotrifluoromethylpyridne derivatives ISHIHARA SANGYO KAISHA, LTD. (JP) 2003-06-12 US claimed
EP-1252889-A1 REMEDIES OR PREVENTIVES FOR PULMONARY INSUFFICIENCY CONTAINING DIAMINOTRIFLUOROMETHYLPYRIDINE DERIVATIVES ISHIHARA SANGYO KAISHA, LTD. (JP) 2002-10-30 EP claimed
EP-0228846-B1 AMINO-TRIFLUOROMETHYLPYRIDINE COMPOUND AND PROCESS FOR PREPARING THE SAME ISHIHARA SANGYO KAISHA, LTD. (JP) 1992-04-22 EP claimed
US-4762928-A PESTICIDES, MEDICINES ISHIHARA SANGYO KAISHA LTD. (JP) 1988-08-09 US claimed
EP-0228846-A1 Amino-trifluoromethylpyridine compound and process for preparing the same ISHIHARA SANGYO KAISHA, LTD. (JP) 1987-07-15 EP claimed
JP-62155259-A None JP disclosed
JP-6247934-A None JP disclosed
EP-4727932-A1 SMALL MOLECULE LIGANDS AND APTAMERS MeiraGTx Gene Regulation Limited (GB) 2026-04-22 EP disclosed
US-20260098047-A1 Anti-Giardial Compounds COMMW SCIENT IND RES ORG (AU) 2026-04-09 US disclosed
EP-4720060-A1 PRMT5 INHIBITORS Ryvu Therapeutics S.A. (PL) 2026-04-08 EP disclosed
US-4731450-A Process for perfluoroalkylation of aromatic derivatives RHONE-POULENC SPECIALITES CHIMIQUES (FR) 1988-03-15 US disclosed
EP-0228846-A1 Amino-trifluoromethylpyridine compound and process for preparing the same ISHIHARA SANGYO KAISHA, LTD. (JP) 1987-07-15 EP disclosed
EP-0228846-A1 Amino-trifluoromethylpyridine compound and process for preparing the same ISHIHARA SANGYO KAISHA, LTD. (JP) 1987-07-15 EP disclosed
EP-0228846-A1 Amino-trifluoromethylpyridine compound and process for preparing the same ISHIHARA SANGYO KAISHA, LTD. (JP) 1987-07-15 EP disclosed
JP-S62155259-A AMINOTRIFLUOROMETHYLPYRIDINE AND ITS PRODUCTION ISHIHARA SANGYO KAISHA LTD 1987-07-10 JP disclosed
EP-0206951-A2 Process for the perfluoroalkylation of aromatic derivatives RHONE-POULENC CHIMIE (FR) 1986-12-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030109551-A1 Remedies or preventives for pulmonary insufficiency containing diaminotrifluoromethylpyridne derivatives CBR1, CBR3, WDR1 HTT 4289/4885HSD17B10 2161/4885KDM4E 3997/4885
US-20260098047-A1 Anti-Giardial Compounds GNAO1, GPR6, MGAT3 HTT 3585/4885HSD17B10 2925/4885KDM4E 3910/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.