SCHEMBL1026306

SCHEMBL1026306

COc1cccnc1N1CCNCC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.57
HTR3E A5X5Y0 1/20 0.57
HTR3B O95264 1/20 0.57
ADRB1 P08588 1/20 0.57
DRD2 P14416 1/20 0.57
DRD3 P35462 1/20 0.57
HTR3A P46098 1/20 0.57
HTR6 P50406 1/20 0.57
HTR3D Q70Z44 1/20 0.57
HTR3C Q8WXA8 1/20 0.57
SIGMAR1 Q99720 1/20 0.57
LMNA P02545 1/20 0.55
MAPT P10636 1/20 0.55
EPHX2 P34913 1/20 0.55
SLC2A1 P11166 1/20 0.52
SLC2A2 P11168 1/20 0.52
SLC2A3 P11169 1/20 0.52
HTR7 P34969 2/20 0.51
HTR1A P08908 1/20 0.50
SLC6A2 P23975 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1969103 0.98 LMNA (0.58) CYP2C19HTR3EHTR3BADRB1DRD2
Hydrochloric Acid SCHEMBL30069211 0.98 LMNA (0.58) CYP2C19HTR3EHTR3BADRB1DRD2
Hydrochloric Acid SCHEMBL26600676 0.98 LMNA (0.58) CYP2C19HTR3EHTR3BADRB1DRD2
Hydrochloric Acid SCHEMBL30069213 0.98 LMNA (0.58) CYP2C19HTR3EHTR3BADRB1DRD2
SCHEMBL12986602 0.94 HTR3A (0.51) CYP2C19HTR3EHTR3BADRB1DRD2
Hydrochloric Acid SCHEMBL1063578 0.93 LMNA (0.52) CYP2C19HTR3EHTR3BADRB1DRD2
SCHEMBL30585959 0.85 SLC2A1 (0.52) CYP2C19DRD2DRD3MAPTSLC2A1
SCHEMBL29086088 0.85 SLC2A1 (0.52) CYP2C19DRD2DRD3MAPTSLC2A1
SCHEMBL15533598 0.84 EPHX2 (0.52) EPHX2HTR1ASLC6A2ALDH1A1
SCHEMBL31652008 0.84 EPHX2 (0.49) CYP2C19HTR3EHTR3BADRB1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 92 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250214977-A1 STAT6 INHIBITORS AND USES THEREOF KYMERA THERAPEUTICS, INC. 2025-07-03 US disclosed
US-20230340011-A1 STEROIDAL COMPOSITIONS AND METHODS OF TREATING LIPOGENIC CANCERS Asteroid Therapeutics 2023-10-26 US disclosed
US-20230340011-A1 STEROIDAL COMPOSITIONS AND METHODS OF TREATING LIPOGENIC CANCERS Asteroid Therapeutics 2023-10-26 US disclosed
CN-112154145-B Piperazine azaspiro derivatives 辉瑞大药厂 2023-10-17 CN disclosed
EP-4219464-A1 PIPERAZINE AZASPIRO DERIVAVES Pfizer Inc. (US) 2023-08-02 EP disclosed
EP-4219464-A1 PIPERAZINE AZASPIRO DERIVAVES Pfizer Inc. (US) 2023-08-02 EP disclosed
US-20230192654-A1 PIPERAZINE AZASPIRO DERIVATIVES PFIZER INC. 2023-06-22 US disclosed
US-20230192654-A1 PIPERAZINE AZASPIRO DERIVATIVES PFIZER INC. 2023-06-22 US disclosed
US-20230192654-A1 PIPERAZINE AZASPIRO DERIVATIVES PFIZER INC. 2023-06-22 US disclosed
EP-3768669-B1 PIPERAZINE AZASPIRO DERIVAVES PFIZER (US) 2023-01-25 EP disclosed
EP-0645385-A1 Antimigraine cyclobutenedione derivatives of indolylalkyl-pyridinyl and pyrimidinylpiperazines Bristol-Myers Squibb Company (US) 1995-03-29 EP disclosed
EP-0345808-B1 1-Indolylalkyl-4-(substituted-pyridinyl)piperazines BRISTOL MYERS SQUIBB CO (US) 1995-01-11 EP disclosed
US-4954502-A Antidepressants BRISTOL-MYERS SQUIBB COMPANY (US) 1990-09-04 US disclosed
EP-0200968-B1 SUCCINIMIDE DERIVATIVES, THEIR PRODUCTION AND USE SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1990-08-29 EP disclosed
EP-0345808-A1 1-Indolylalkyl-4-(substituted-pyridinyl)piperazines Bristol-Myers Squibb Company (US) 1989-12-13 EP disclosed
US-4843078-A ANXIOLYTIC AGENTS SUMITONO PHARMACEUTICAL COMPANY, LIMITED (JP) 1989-06-27 US disclosed
US-4757073-A Antipsychotic agents BRISTOL-MYERS COMPANY (US) 1988-07-12 US disclosed
EP-0200968-A1 Succinimide derivatives, their production and use SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1986-11-12 EP disclosed
US-4619930-A Antipsychotic cyclic imide derivatives of 2-(4-butylpiperazin-1-yl)pyridines, compositions and use BRISTOL-MYERS COMPANY (US) 1986-10-28 US disclosed
US-4305944-A TRANQUILIZERS, NEUROLEPTIC AGENTS MEAD JOHNSON & COMPANY (US) 1981-12-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230192654-A1 PIPERAZINE AZASPIRO DERIVATIVES CHRM1, CHRM2, CHRM5 CYP2C19 502/4885HTR3E 1289/4885HTR3B 479/4885
US-20230340011-A1 STEROIDAL COMPOSITIONS AND METHODS OF TREATING LIPOGENIC CANCERS SREBF1, SREBF2, NR1H3 CYP2C19 2761/4885HTR3E 4256/4885HTR3B 3634/4885
US-20250214977-A1 STAT6 INHIBITORS AND USES THEREOF STAT6, STAT5B, STAT5A CYP2C19 4391/4885HTR3E 2136/4885HTR3B 2505/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.