SCHEMBL10269012

SCHEMBL10269012

Cc1c[nH]c2ncc(N)cc12

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MET P08581 1/20 0.43
PRMT5 O14744 1/20 0.42
WDR77 Q9BQA1 1/20 0.42
BTK Q06187 6/20 0.41
ITK Q08881 6/20 0.41
NTRK1 P04629 5/20 0.40
GSK3B P49841 1/20 0.40
KIT P10721 4/20 0.40
MAP3K11 Q16584 1/20 0.39
CLK1 P49759 1/20 0.38
DYRK1A Q13627 1/20 0.38
DYRK2 Q92630 1/20 0.38
DYRK1B Q9Y463 1/20 0.38
PIK3CA P42336 1/20 0.37
AXL P30530 1/20 0.37
PRKCI P41743 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7921128 0.80 MET (0.46) METPRMT5WDR77BTKITK
SCHEMBL14883424 0.77 JAK2 (0.54) METPRMT5WDR77BTKITK
SCHEMBL1566306 0.77 ITK (0.54) METPRMT5WDR77BTKITK
SCHEMBL25841381 0.77 MET (0.43) METPRMT5WDR77BTKITK
SCHEMBL14041214 0.77 MET (0.43) METPRMT5WDR77BTKITK
SCHEMBL24005850 0.77 PRMT5 (0.42) PRMT5WDR77BTKITKNTRK1
SCHEMBL25971496 0.77 BRD4 (0.47) NTRK1GSK3BKITMAP3K11CLK1
SCHEMBL1774189 0.77 NTRK1 (0.38) PRMT5WDR77NTRK1GSK3BKIT
SCHEMBL1772956 0.77 MAP3K11 (0.39) NTRK1GSK3BKITMAP3K11CLK1
SCHEMBL10212537 0.77 PRMT5 (0.45) PRMT5WDR77NTRK1GSK3BKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8338452-B2 Raf inhibitor compounds and methods of use thereof ARRAY BIOPHARMA INC. (US) 2012-12-25 US disclosed
US-20120053345-A1 Indazole Compounds ABBOTT LABORATORIES (US) 2012-03-01 US disclosed
US-8008481-B2 Indazole compounds ABBVIE INC. 2011-08-30 US disclosed
US-20110110889-A1 RAF INHIBITOR COMPOUNDS AND METHODS OF USE THEREOF Array Bio Pharma Inc. (US) 2011-05-12 US disclosed
US-20070282101-A1 Indazole compounds ABBVIE INC. 2007-12-06 US disclosed
WO-2007117465-A2 INDAZOLE COMPOUNDS ABBOTT LABORATORIES (US) 2007-10-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070282101-A1 Indazole compounds CYP3A43, CYP3A7, UGT1A1 MET 2464/4885PRMT5 1613/4885WDR77 3008/4885
US-20110110889-A1 RAF INHIBITOR COMPOUNDS AND METHODS OF USE THEREOF BRAF, RAF1, ARAF MET 542/4885PRMT5 2445/4885WDR77 2667/4885
US-20120053345-A1 Indazole Compounds CYP3A43, CYP3A7, UGT1A1 MET 2464/4885PRMT5 1613/4885WDR77 3008/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.