SCHEMBL10285346

SCHEMBL10285346

NCc1cc(O)c(O)cn1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RECQL P46063 6/20 0.33
TDP1 Q9NUW8 6/20 0.33
MAPT P10636 5/20 0.33
APEX1 P27695 4/20 0.33
BLM P54132 4/20 0.33
KDM4E B2RXH2 4/20 0.33
MAPK1 P28482 4/20 0.33
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
ADRA2A P08913 3/20 0.33
DRD2 P14416 3/20 0.33
DRD1 P21728 3/20 0.33
HPGD P15428 2/20 0.33
THRB P10828 2/20 0.33
RAD52 P43351 2/20 0.33
ADRB2 P07550 2/20 0.33
ADRA1D P25100 2/20 0.33
ADRA1A P35348 2/20 0.33
ADRA1B P35368 2/20 0.33
TAAR1 Q96RJ0 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3568446 0.82 KDM4E (0.34) MAPTKDM4EMEN1KMT2ACYP3A4
SCHEMBL13343544 0.80 NOS3 (0.35) MAPTKDM4EMAPK1HPGDLMNA
SCHEMBL14001672 0.80
SCHEMBL9197728 0.78
SCHEMBL10285565 0.78 ALDH1A1 (0.39) ALDH1A1
SCHEMBL10285300 0.76 TRPA1 (0.38) ALOX15
SCHEMBL3567972 0.76 NFKB1 (0.42) APEX1BLMMAPK1MEN1KMT2A
SCHEMBL3565806 0.74 BACE1 (0.47) MAPTKMT2AHPGDLMNAHSD17B10
SCHEMBL3573538 0.72 CSNK2A1 (0.41) TDP1MAPTKDM4EMEN1KMT2A
SCHEMBL19700919 0.71 ESR1 (0.34) TDP1MAPTKDM4EHPGDALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2468743-A1 Nitrogen-containing bicyclic compounds useful as antibacterial agents Toyama Chemical Co., Ltd. (JP) 2012-06-27 EP disclosed
EP-1900732-A1 NOVEL NITROGENATED HETEROCYCLIC COMPOUND AND SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2008-03-19 EP disclosed
WO-2007065288-A2 USEFUL COMBINATIONS OF MONOBACTAM ANTIBIOTICS WITH BETA-LACTAMASE INHIBITORS BASILEA PHARMACEUTICA AG (CH) 2007-06-14 WO disclosed