SCHEMBL10292467

SCHEMBL10292467

CC(C)(C)OC(=O)N1CCCC(c2nc3ccc(Cl)nc3[nH]2)C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 2/20 0.50
JAK2 O60674 1/20 0.45
JAK1 P23458 1/20 0.45
GRIN2B Q13224 2/20 0.43
HCAR1 Q9BXC0 1/20 0.43
CHEK2 O96017 2/20 0.43
PARP1 P09874 1/20 0.43
TRPV3 Q8NET8 1/20 0.43
CYP2C9 P11712 1/20 0.42
PRMT5 O14744 2/20 0.41
MAPK1 P28482 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GLA P06280 1/20 0.41
HPGD P15428 1/20 0.41
RECQL P46063 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PBK Q96KB5 1/20 0.40
USP30 Q70CQ3 1/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29657985 0.82 HPGDS (0.47) HPGDSHCAR1CHEK2PARP1TRPV3
SCHEMBL22701135 0.82 HPGDS (0.47) HPGDSHCAR1CHEK2PARP1TRPV3
SCHEMBL742218 0.81 HPGDS (0.52) HPGDSJAK2JAK1GRIN2BHCAR1
SCHEMBL742219 0.81 HPGDS (0.52) HPGDSJAK2JAK1GRIN2BHCAR1
SCHEMBL16584386 0.81 DGAT2 (0.57) HPGDS
SCHEMBL16584385 0.81 DGAT2 (0.57) HPGDS
SCHEMBL16584388 0.81 DGAT2 (0.57) HPGDS
SCHEMBL19408169 0.80 HPGDS (0.57) HPGDSPARP1CYP2C9PRMT5MAPK1
SCHEMBL739188 0.80 HPGDS (0.57) HPGDSPARP1CYP2C9PRMT5MAPK1
SCHEMBL762565 0.80 HPGDS (0.57) HPGDSPARP1CYP2C9PRMT5MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed