SCHEMBL1029403

SCHEMBL1029403

COc1cccc(CCNC(=O)c2c(-c3ccc(C)cc3)c(C)cn2C)c1OC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.45
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA14 Q9ULX7 1/20 0.42
ROCK2 O75116 1/20 0.41
ROCK1 Q13464 1/20 0.41
HPGD P15428 4/20 0.41
MAPT P10636 3/20 0.40
TP53 P04637 3/20 0.40
PARP1 P09874 1/20 0.40
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
GAA P10253 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
LMNA P02545 3/20 0.39
ALDH1A1 P00352 3/20 0.39
ATM Q13315 2/20 0.39
KDM4E B2RXH2 2/20 0.39
HSD17B10 Q99714 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1031789 0.90 ROCK2 (0.52) NAMPTROCK2ROCK1HPGDMAPT
SCHEMBL1030186 0.77 GAA (0.46) ROCK2ROCK1HPGDTP53GAA
SCHEMBL1030747 0.76 NPC1 (0.53) HPGDMAPTTP53SMN1; SMN2
SCHEMBL17150039 0.72 CA12 (0.61) NAMPTCA12CA1CA2CA14
SCHEMBL1081685 0.71 NPSR1 (0.60) L3MBTL1ALDH1A1TSHR
SCHEMBL1028545 0.71 ROCK2 (0.48) NAMPTROCK2ROCK1HPGDMAPT
SCHEMBL1009815 0.71 MTNR1A (0.75) CA12CA1CA2CA14MTNR1A
SCHEMBL1032372 0.71 TP53 (0.54) HPGDMAPTTP53GAAL3MBTL1
SCHEMBL19055872 0.70 CA12 (0.56) NAMPTCA12CA1CA2CA14
SCHEMBL1029749 0.70 NPC1 (0.47) HPGDMAPTTP53GAAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035375-B1 1,3-DISUBSTITUTED 4-METHYL-1H-PYRROLE-2-CARBOXAMIDES AND THEIR USE FOR THE MANUFACTURE OF MEDICAMENTS GRUENENTHAL GMBH (DE) 2011-01-19 EP claimed