SCHEMBL1081685

SCHEMBL1081685

Cc1ccc(-c2c(C)cn(C)c2C(=O)NCCN2CCCC2)cc1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.60
KMT2A Q03164 4/20 0.48
MEN1 O00255 3/20 0.47
CACNA1G O43497 2/20 0.45
ALDH1A1 P00352 3/20 0.45
CYP2D6 P10635 2/20 0.45
TSHR P16473 2/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C19 P33261 1/20 0.45
POLB P06746 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
GLA P06280 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
RECQL P46063 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1030647 0.83 HTT (0.59) KMT2AALDH1A1TSHRL3MBTL1RECQL
SCHEMBL1031916 0.83 NPSR1 (0.51) NPSR1CACNA1GTSHR
SCHEMBL1031140 0.81 NPSR1 (0.49) NPSR1KMT2AMEN1CACNA1GALDH1A1
SCHEMBL1031613 0.81 ALDH1A1 (0.61) ALDH1A1TSHRPOLB
SCHEMBL1031841 0.80 NPSR1 (0.47) NPSR1KMT2AMEN1CACNA1GALDH1A1
SCHEMBL1028264 0.77 CACNA1G (0.47) NPSR1KMT2AMEN1CACNA1G
SCHEMBL279945 0.76 NPSR1 (0.97) NPSR1KMT2AMEN1CACNA1GALDH1A1
SCHEMBL1030747 0.76 NPC1 (0.53) KMT2A
SCHEMBL10195008 0.75 NPSR1 (0.94) NPSR1KMT2AMEN1CACNA1GALDH1A1
SCHEMBL1031804 0.73 ALDH1A1 (0.42) KMT2AMEN1ALDH1A1POLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035375-B1 1,3-DISUBSTITUTED 4-METHYL-1H-PYRROLE-2-CARBOXAMIDES AND THEIR USE FOR THE MANUFACTURE OF MEDICAMENTS GRUENENTHAL GMBH (DE) 2011-01-19 EP claimed