SCHEMBL10313571

SCHEMBL10313571

CCOC(=O)c1c(O)[nH]c2c(-c3ccc(C)cc3)c(CC)nn2c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
ALDH1A1 P00352 6/20 0.39
MAPT P10636 2/20 0.39
PKM P14618 1/20 0.39
PLAT P00750 1/20 0.38
CACNB4 O00305 1/20 0.38
CACNA1A O00555 1/20 0.38
CACNA1G O43497 1/20 0.38
CACNG3 O60359 1/20 0.38
CACNA1F O60840 1/20 0.38
CACNA1H O95180 1/20 0.38
ACHE P22303 1/20 0.38
CACNB3 P54284 1/20 0.38
CACNA2D1 P54289 1/20 0.38
CACNG7 P62955 1/20 0.38
CACNA1B Q00975 1/20 0.38
CACNA1D Q01668 1/20 0.38
CACNB1 Q02641 1/20 0.38
CACNG1 Q06432 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10313456 0.89 MAPT (0.44) CYP1A2CYP2C19ALDH1A1MAPTPKM
SCHEMBL10275766 0.89 MAPT (0.43) CYP1A2CYP2C19ALDH1A1MAPTPLAT
SCHEMBL10313580 0.85 MAT2A (0.50) ALDH1A1MAPTPLATKDM4EGAA
SCHEMBL10313590 0.81 MAPT (0.52) CYP1A2CYP2C19ALDH1A1MAPTPLAT
SCHEMBL10275637 0.80 ALOX5 (0.37) CYP1A2CYP2C19ALDH1A1MAPTPLAT
SCHEMBL10275627 0.80 MAPT (0.41) CYP1A2ALDH1A1MAPTPLATHTT
SCHEMBL10276177 0.78 MAPT (0.44) ALDH1A1MAPTPLATHTTKDM4E
SCHEMBL10275451 0.75 MAT2A (0.47) ALDH1A1MAPTPLATKDM4EGAA
SCHEMBL10313511 0.74 GPR119 (0.43) ALDH1A1MAPTPLATHTTKDM4E
SCHEMBL10313493 0.74 SLC34A1 (0.43) ALDH1A1MAPTPLATHTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120178915-A1 PYRIMIDINE DERIVATIVES AND ANALOGS, PREPARATION METHOD AND USE THEREOF XU LIFENG (US) 2012-07-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120178915-A1 PYRIMIDINE DERIVATIVES AND ANALOGS, PREPARATION METHOD AND USE THEREOF TYMP, TYMS, ADORA3 CYP1A2 108/4885CYP2C19 620/4885ALDH1A1 572/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.