SCHEMBL10313595

SCHEMBL10313595

CC1=NN2C(=O)C=C(c3ccc(C#N)cc3)NC2C=C1c1ccccc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
SLC11A2 P49281 1/20 0.34
CGAS Q8N884 1/20 0.32
ALDH1A1 P00352 1/20 0.32
IDO1 P14902 1/20 0.32
GABRA1 P14867 1/20 0.31
GABRG2 P18507 1/20 0.31
GABRB3 P28472 1/20 0.31
GABRA5 P31644 1/20 0.31
GABRA3 P34903 1/20 0.31
GABRA2 P47869 1/20 0.31
CYP11B2 P19099 1/20 0.31
CASP6 P55212 1/20 0.31
AR P10275 1/20 0.31
BRD4 O60885 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
MAOB P27338 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10313496 0.93 ALDH1A1 (0.35) ALDH1A1CYP11B2MAOB
SCHEMBL10275578 0.90 SIRT5 (0.40) AR
SCHEMBL10276240 0.88 KIF11 (0.40) CYP11B2MAOB
SCHEMBL10275313 0.82 KDM4E (0.35) MEN1KMT2ABRD4
SCHEMBL10275367 0.78 ALOX5AP (0.35) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL10313719 0.75 CNR2 (0.34)
SCHEMBL10276245 0.74 NR3C2 (0.38) AR
SCHEMBL10275787 0.73 ALOX5AP (0.34) GABRG2GABRB3GABRA5GABRA3AR
SCHEMBL10276334 0.72 KIF11 (0.39) CYP11B2MAOB
SCHEMBL10276332 0.72 KIF11 (0.39) CYP11B2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120178915-A1 PYRIMIDINE DERIVATIVES AND ANALOGS, PREPARATION METHOD AND USE THEREOF XU LIFENG (US) 2012-07-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120178915-A1 PYRIMIDINE DERIVATIVES AND ANALOGS, PREPARATION METHOD AND USE THEREOF TYMP, TYMS, ADORA3 ATM 1770/4885MEN1 4229/4885KMT2A 4649/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.