SCHEMBL10313630

SCHEMBL10313630

[C-]#[N+]c1ccc(-n2cnc3c(N)nc(-c4ccc(F)cc4F)nc32)cc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PI4KA P42356 6/20 0.40
PI4K2B Q8TCG2 6/20 0.40
PI4K2A Q9BTU6 6/20 0.40
PI4KB Q9UBF8 6/20 0.40
CFTR P13569 2/20 0.39
MAPK14 Q16539 4/20 0.38
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
CYP17A1 P05093 1/20 0.34
EGFR P00533 1/20 0.33
KIF5C O60282 1/20 0.33
KIF11 P52732 1/20 0.33
KIF5A Q12840 1/20 0.33
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
XDH P47989 3/20 0.32
GRM1 Q13255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10313636 0.89 MAPK14 (0.36) PI4KAPI4K2BPI4K2API4KBCFTR
SCHEMBL10276251 0.83 PI4KA (0.40) PI4KAPI4K2BPI4K2API4KBCFTR
SCHEMBL10313633 0.77 XDH (0.42) PTGS1PTGS2XDH
SCHEMBL10313642 0.77 CYP17A1 (0.38) PI4KAPI4K2BPI4K2API4KBCYP17A1
SCHEMBL10313629 0.76 PI4KA (0.41) PI4KAPI4K2BPI4K2API4KBCFTR
SCHEMBL10313898 0.72 CTSV (0.39) MAPK14PTGS1PTGS2KIF5CKIF11
SCHEMBL27870411 0.70 CFTR (0.49) PI4KAPI4K2BPI4K2API4KBCFTR
SCHEMBL10313616 0.65 PI4KA (0.32) PI4KAPI4K2BPI4K2API4KB
SCHEMBL6493961 0.61 MAPK14 (0.62) MAPK14ADORA1
SCHEMBL10275806 0.60 XDH (0.42) PTGS1PTGS2XDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120178915-A1 PYRIMIDINE DERIVATIVES AND ANALOGS, PREPARATION METHOD AND USE THEREOF XU LIFENG (US) 2012-07-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120178915-A1 PYRIMIDINE DERIVATIVES AND ANALOGS, PREPARATION METHOD AND USE THEREOF TYMP, TYMS, ADORA3 PI4KA 2350/4885PI4K2B 3385/4885PI4K2A 3326/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.