SCHEMBL1031580

SCHEMBL1031580

Cc1cn(C)c(C(=O)NCc2ccccn2)c1-c1ccco1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.55
L3MBTL1 Q9Y468 6/20 0.53
HPGD P15428 4/20 0.53
KDM4E B2RXH2 4/20 0.53
MAPT P10636 3/20 0.53
POLB P06746 2/20 0.53
KMT2A Q03164 2/20 0.53
MEN1 O00255 1/20 0.53
THRB P10828 1/20 0.53
PKM P14618 1/20 0.53
ALOX15 P16050 1/20 0.53
NR4A1 P22736 1/20 0.53
APEX1 P27695 1/20 0.53
CASP1 P29466 1/20 0.53
PTPN7 P35236 1/20 0.53
RECQL P46063 1/20 0.53
BLM P54132 1/20 0.53
CASP7 P55210 1/20 0.53
MCL1 Q07820 1/20 0.53
ESR2 Q92731 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1031424 0.79 ALDH1A1 (0.48) ALDH1A1L3MBTL1KDM4EMAPTPOLB
SCHEMBL1031918 0.76 ALDH1A1 (0.47) ALDH1A1L3MBTL1HPGDKDM4EMAPT
SCHEMBL1030582 0.76 MEN1 (0.47) L3MBTL1KDM4EMAPTPOLBKMT2A
SCHEMBL1032220 0.75 RAB9A (0.47) ALDH1A1L3MBTL1HPGDKDM4EMAPT
SCHEMBL1032676 0.75 ADORA3 (0.49) ALDH1A1L3MBTL1HPGDKDM4EMAPT
SCHEMBL1032230 0.75 ADORA3 (0.55) ALDH1A1L3MBTL1HPGDKDM4EPOLB
SCHEMBL1031541 0.74 RAB9A (0.53) ALDH1A1HPGDMAPTPOLBKMT2A
SCHEMBL1030274 0.73 POLB (0.46) ALDH1A1L3MBTL1HPGDKDM4EMAPT
SCHEMBL1033134 0.73 P2RX7 (0.43) SMN1; SMN2
SCHEMBL1475078 0.72 NPC1 (0.72) ALDH1A1L3MBTL1HPGDKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035375-B1 1,3-DISUBSTITUTED 4-METHYL-1H-PYRROLE-2-CARBOXAMIDES AND THEIR USE FOR THE MANUFACTURE OF MEDICAMENTS GRUENENTHAL GMBH (DE) 2011-01-19 EP claimed