SCHEMBL10317472

SCHEMBL10317472

Cc1ccc(-n2ccc3cc(NC(C(=O)O)S(=O)(=O)c4cc(Cl)cc(Cl)c4)ccc32)nn1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACLY P53396 1/20 0.35
ROCK1 Q13464 2/20 0.32
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32
APH1B Q8WW43 1/20 0.32
NCSTN Q92542 1/20 0.32
APH1A Q96BI3 1/20 0.32
PSENEN Q9NZ42 1/20 0.32
PHGDH O43175 3/20 0.31
PIM1 P11309 1/20 0.31
CSNK2A1 P68400 1/20 0.31
PIM3 Q86V86 1/20 0.31
PIM2 Q9P1W9 1/20 0.31
HTR2C P28335 1/20 0.31
IRAK4 Q9NWZ3 1/20 0.31
RORC P51449 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10319470 0.87 PHGDH (0.31) ROCK1PHGDH
SCHEMBL10321256 0.85 ROCK1 (0.37) ACLYROCK1PSEN1PSEN2APH1B
SCHEMBL3300353 0.74 ACLY (0.31) ACLY
SCHEMBL3300118 0.74 DGAT1 (0.32) ACLY
SCHEMBL3301072 0.73 KEAP1 (0.39)
SCHEMBL3294583 0.73 CKS1B (0.40)
SCHEMBL15712556 0.72 MEN1 (0.43)
SCHEMBL3298512 0.71 UTS2R (0.33) ACLY
SCHEMBL2967385 0.71 CYP3A4 (0.42) ACLYPSEN1PSEN2APH1BNCSTN
SCHEMBL3021252 0.70 S1PR1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121600-B1 SUBSTITUTED ARYLSULPHONYLGLYCINES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS BOEHRINGER INGELHEIM INT (DE) 2012-07-18 EP claimed