SCHEMBL10337992

SCHEMBL10337992

C=CCc1ccc2ccc3cccc4c(OC)cc1c2c34

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
PPARG P37231 3/20 0.40
PPARD Q03181 2/20 0.40
PPARA Q07869 2/20 0.40
ELANE P08246 1/20 0.39
ALOX5 P09917 2/20 0.38
GABRA1 P14867 1/20 0.38
CNR2 P34972 1/20 0.38
GABRB2 P47870 1/20 0.38
RXRA P19793 1/20 0.38
KDM4E B2RXH2 3/20 0.38
GAA P10253 2/20 0.38
CYP3A4 P08684 2/20 0.38
ALOX15 P16050 1/20 0.38
AR P10275 1/20 0.37
PTGS1 P23219 1/20 0.37
TRPM8 Q7Z2W7 1/20 0.37
MAPT P10636 3/20 0.37
TDP1 Q9NUW8 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28804419 0.81 HSD17B10 (0.44) ALDH1A1GABRA1GABRB2KDM4EGAA
SCHEMBL7749583 0.78 GABRA1 (0.41) ALDH1A1GABRA1GABRB2KDM4EGAA
SCHEMBL728402 0.76 KMT2A (0.47) ALDH1A1GABRA1GABRB2KDM4ECYP3A4
SCHEMBL8724008 0.75 ALDH1A1 (0.43) ALDH1A1GABRA1GABRB2KDM4ECYP3A4
SCHEMBL16241709 0.74 CYP1A2 (0.52) ALDH1A1PPARGPPARDPPARARXRA
SCHEMBL729571 0.73 ALDH1A1 (0.47) ALDH1A1GABRA1GABRB2KDM4ECYP3A4
SCHEMBL27930641 0.72 ALDH1A1 (0.55) ALDH1A1GABRA1GABRB2KDM4ECYP3A4
SCHEMBL5748760 0.72 IDO1 (0.50) ALDH1A1PPARGPPARDPPARARXRA
SCHEMBL28831011 0.72 ALDH1A1 (0.45) ALDH1A1GABRA1GABRB2KDM4ECYP3A4
SCHEMBL4338851 0.72 MEN1 (0.37) ALDH1A1GABRA1GABRB2KDM4ECYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0365539-A4 HUMAN LEUCOCYTE ELASTASE INHIBITOR COMPOUNDS 1990-12-05 EP disclosed
EP-0365539-A1 HUMAN LEUCOCYTE ELASTASE INHIBITOR COMPOUNDS AUSTRALIAN COMMERCIAL RESEARCH & DEVELOPMENT LIMITED (AU) 1990-05-02 EP disclosed
WO-1988010258-A1 HUMAN LEUCOCYTE ELASTASE INHIBITOR COMPOUNDS LA TROBE UNIVERSITY (AU) 1988-12-29 WO disclosed