SCHEMBL5748760

SCHEMBL5748760

COc1cc2c(N)ccc3ccc4cccc1c4c32

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.50
EP300 Q09472 2/20 0.49
KAT8 Q9H7Z6 1/20 0.49
PPARG P37231 2/20 0.43
RXRA P19793 1/20 0.43
PPARD Q03181 1/20 0.43
PPARA Q07869 1/20 0.43
MAPT P10636 1/20 0.42
MCHR1 Q99705 1/20 0.41
ALDH1A1 P00352 5/20 0.41
HSD17B10 Q99714 3/20 0.41
HPGD P15428 2/20 0.41
CYP1A2 P05177 2/20 0.41
THRB P10828 1/20 0.41
CYP3A4 P08684 3/20 0.40
TSHR P16473 2/20 0.40
APP P05067 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
NQO1 P15559 1/20 0.40
KEAP1 Q14145 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5746447 0.90 IDO1 (0.47) IDO1EP300KAT8PPARGRXRA
SCHEMBL5748942 0.83 IDO1 (0.43) IDO1EP300KAT8PPARGRXRA
SCHEMBL16241709 0.82 CYP1A2 (0.52) PPARGRXRAPPARDPPARAMAPT
SCHEMBL5748372 0.80 CYP1A2 (0.43) IDO1EP300PPARGRXRAPPARD
SCHEMBL5750461 0.79 ALDH1A1 (0.42) IDO1EP300KAT8PPARGRXRA
SCHEMBL5749544 0.78 IDO1 (0.57) IDO1EP300KAT8PPARGMAPT
SCHEMBL5746648 0.78 IDO1 (0.57) IDO1EP300KAT8PPARGMAPT
SCHEMBL5750998 0.77 ALDH1A1 (0.53) MAPTALDH1A1HSD17B10HPGDCYP1A2
SCHEMBL5747739 0.75 CYP1A2 (0.41) PPARGRXRAPPARDPPARAMAPT
SCHEMBL426014 0.74 ALDH1A1 (0.48) IDO1EP300KAT8MAPTMCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060293503-A1 Polyaminopyridines and method for producing same SUMITOMO SEIKA CHEMICALS CO., LTD (JP) 2006-12-28 US disclosed
EP-1669390-A1 POLYAMINOPYRIDINES AND METHOD FOR PRODUCING SAME SUMITOMO SEIKA CHEMICALS CO., LTD. (JP) 2006-06-14 EP disclosed