SCHEMBL10340263

SCHEMBL10340263

O=[N+]([O-])C1Cc2c[nH]c3ccc(O)c(c23)C1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.44
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
HTR1A P08908 1/20 0.36
HTR2A P28223 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10340259 0.80 MTNR1A (0.57) MTNR1AMTNR1BHTR1AHTR2A
SCHEMBL23248790 0.77 MEN1 (0.40)
SCHEMBL10340613 0.75 MAOA (0.48) MAOAMTNR1AMTNR1BHTR1A
SCHEMBL10682096 0.69
SCHEMBL6996649 0.61 CYP3A4 (0.39) HTR1AHTR2A
SCHEMBL13701016 0.60 MCL1 (0.41) MAOAMTNR1AMTNR1B
Hyrtioreticulin D SCHEMBL30434518 0.59 HTR2A (0.39) MAOAMTNR1AMTNR1BHTR1AHTR2A
SCHEMBL23261875 0.57 MAP3K14 (0.39) MAOAMTNR1AMTNR1BHTR1A
SCHEMBL23261947 0.57 DRD2 (0.38) MAOAMTNR1AMTNR1BHTR1AHTR2A
SCHEMBL4420013 0.57 HTR2C (0.39) MAOAHTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0162695-A1 6-Oxygenated-1,3,,4,5-Tetrahydrobenz(cd)indol-4-amines SMITHKLINE BEECHAM CORPORATION (US) 1985-11-27 EP claimed
EP-0162695-B1 6-OXYGENATED-1,3,,4,5-TETRAHYDROBENZ(CD)INDOL-4-AMINES SMITHKLINE BEECHAM CORPORATION (US) 1990-01-17 EP disclosed
EP-0162695-A1 6-Oxygenated-1,3,,4,5-Tetrahydrobenz(cd)indol-4-amines SMITHKLINE BEECHAM CORPORATION (US) 1985-11-27 EP disclosed