SCHEMBL10345289

SCHEMBL10345289

COCCc1ccc(C(OC(c2ccc(CCOC)cc2)C2CO2)C2CO2)cc1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.36
ACACA Q13085 1/20 0.36
NR3C1 P04150 1/20 0.33
ADRB2 P07550 1/20 0.33
ADRB1 P08588 1/20 0.33
CYP2D6 P10635 1/20 0.33
ADRA1A P35348 1/20 0.33
CYP2J2 P51589 1/20 0.33
PDE4D Q08499 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ENPP2 Q13822 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11862422 0.91 MEN1 (0.36) L3MBTL1
SCHEMBL9502745 0.81 THRA (0.41)
SCHEMBL3242474 0.80 TSHR (0.40) L3MBTL1
SCHEMBL7871491 0.79 THRA (0.49) ENPP2
SCHEMBL10411867 0.79 THRA (0.49) ENPP2
SCHEMBL27082092 0.79 THRA (0.49) ENPP2
SCHEMBL11507345 0.77 KCNH2 (0.32)
SCHEMBL14889733 0.77 LTA4H (0.32)
SCHEMBL333671 0.75 CA12 (0.41) CYP2D6L3MBTL1
SCHEMBL3784692 0.74 CHRNA7 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0193228-B1 PROCESS FOR PRODUCING OF 4-(2-METHOXYETHYL)-PHENYLGLYCIDYL ETHER AND/OR METOPROLOL GIST-BROCADES N.V. (NL) 1989-11-02 EP claimed
CN-86100965-A Produce 4-(2-methoxyethyl)-phenylglycidyl ether and (or) method of metoprolol 1986-10-01 CN claimed
EP-0193228-A1 Process for producing of 4-(2-methoxyethyl)-phenylglycidyl ether and/or metoprolol GIST-BROCADES N.V. (NL) 1986-09-03 EP claimed
JP-61254194-A None JP disclosed
US-4956284-A Process for producing 4-(2-methoxyethyl)-phenyl-glycidyl ether and/or metoprolol GIST-BROCADES N.V. (NL) 1990-09-11 US disclosed
EP-0193227-B1 PROCESS FOR THE PREPARATION OF ARYLGLYCIDYL ETHERS AND 3-SUBSTITUTED 1-ALKYLAMINO-2-PROPANOLS GIST-BROCADES N.V. (NL) 1990-04-11 EP disclosed
EP-0193228-B1 PROCESS FOR PRODUCING OF 4-(2-METHOXYETHYL)-PHENYLGLYCIDYL ETHER AND/OR METOPROLOL GIST-BROCADES N.V. (NL) 1989-11-02 EP disclosed
EP-0193228-B1 PROCESS FOR PRODUCING OF 4-(2-METHOXYETHYL)-PHENYLGLYCIDYL ETHER AND/OR METOPROLOL GIST-BROCADES N.V. (NL) 1989-11-02 EP disclosed
CN-86102227-A The preparation method of 1-alkylamino-2-propyl alcohol that arylolycidyl ethers and 3-replace 1987-02-04 CN disclosed
JP-S61254194-A PRODUCTION OF 4-(2-METHOXYETHYL)-PHENYLGLYCIDYL ETHER AND/ORMETHOPRROLOLE GIST BROCADES NV 1986-11-11 JP disclosed
CN-86100965-A Produce 4-(2-methoxyethyl)-phenylglycidyl ether and (or) method of metoprolol 1986-10-01 CN disclosed
CN-86100965-A Produce 4-(2-methoxyethyl)-phenylglycidyl ether and (or) method of metoprolol 1986-10-01 CN disclosed
CN-86100965-A Produce 4-(2-methoxyethyl)-phenylglycidyl ether and (or) method of metoprolol 1986-10-01 CN disclosed
EP-0193228-A1 Process for producing of 4-(2-methoxyethyl)-phenylglycidyl ether and/or metoprolol GIST-BROCADES N.V. (NL) 1986-09-03 EP disclosed
EP-0193227-A1 Process for the preparation of arylglycidyl ethers and 3-substituted 1-alkylamino-2-propanols GIST-BROCADES N.V. (NL) 1986-09-03 EP disclosed
EP-0193228-A1 Process for producing of 4-(2-methoxyethyl)-phenylglycidyl ether and/or metoprolol GIST-BROCADES N.V. (NL) 1986-09-03 EP disclosed
EP-0193228-A1 Process for producing of 4-(2-methoxyethyl)-phenylglycidyl ether and/or metoprolol GIST-BROCADES N.V. (NL) 1986-09-03 EP disclosed