SCHEMBL10345596

SCHEMBL10345596

NS(=O)(=O)c1cc2cc(O)ccc2[nH]1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA2 P00918 10/20 1.00
FLT3 P36888 7/20 0.51
PDGFRB P09619 2/20 0.51
ABL1 P00519 1/20 0.51
KIT P10721 1/20 0.51
BCR P11274 1/20 0.51
SMAD3 P84022 1/20 0.50
PDGFRA P16234 1/20 0.45
CLK1 P49759 1/20 0.43
DYRK1A Q13627 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11036272 0.87 CA2 (0.84) CA2FLT3PDGFRBPDGFRA
SCHEMBL10345382 0.86 CA2 (1.00) CA2
SCHEMBL10573479 0.79 CA2 (0.66) CA2
SCHEMBL32681985 0.76 CA2 (1.00) CA2FLT3
SCHEMBL32895 0.76 CA2 (1.00) CA2FLT3
SCHEMBL10345372 0.75 CA2 (1.00) CA2FLT3PDGFRBPDGFRA
SCHEMBL529968 0.71 FLT3 (0.55) CA2FLT3PDGFRBABL1KIT
SCHEMBL830973 0.70 CA2 (0.54) CA2FLT3PDGFRBABL1KIT
SCHEMBL2454392 0.70 FLT3 (0.59) CA2FLT3PDGFRBABL1KIT
SCHEMBL32666155 0.70 FLT3 (0.59) CA2FLT3PDGFRBABL1KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0155214-B1 2-SULFAMOYL-1H-INDOLE DERIVATIVES FOR THE TREATMENT OF ELEVATED INTRAOCULAR PRESSURE MERCK & CO. INC. (US) 1990-03-14 EP disclosed
US-4840963-A FOR GLAUCOMA MERCK & CO., INC. (US) 1989-06-20 US disclosed
EP-0155214-A2 2-sulfamoyl-1H-indole derivatives for the treatment of elevated intraocular pressure MERCK & CO. INC. (US) 1985-09-18 EP disclosed