SCHEMBL10354542

SCHEMBL10354542

c1csc(-c2ccc3scnc3c2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIPK2 O43353 6/20 0.60
RIPK3 Q9Y572 2/20 0.60
KCNH2 Q12809 1/20 0.47
ALDH1A1 P00352 1/20 0.46
HSD17B10 Q99714 1/20 0.46
ALK Q9UM73 1/20 0.45
DYRK1A Q13627 1/20 0.41
KDR P35968 2/20 0.41
TGFBR1 P36897 2/20 0.41
EGFR P00533 1/20 0.41
CYP2E1 P05181 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2A6 P11509 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2B6 P20813 1/20 0.41
LTA4H P09960 1/20 0.41
ERN1 O75460 1/20 0.41
ALOX5AP P20292 1/20 0.40
FEN1 P39748 1/20 0.40
CYP17A1 P05093 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28048502 0.81 ALDH1A1 (0.54) RIPK2RIPK3ALDH1A1HSD17B10DYRK1A
SCHEMBL19579123 0.78 ALDH1A1 (0.44) RIPK2RIPK3ALDH1A1HSD17B10DYRK1A
SCHEMBL29478085 0.77 RIPK2 (0.60) RIPK2RIPK3ALDH1A1HSD17B10DYRK1A
SCHEMBL927048 0.77 RIPK2 (0.60) RIPK2RIPK3ALDH1A1HSD17B10DYRK1A
SCHEMBL22668158 0.75 RIPK2 (0.41) RIPK2RIPK3ALDH1A1HSD17B10DYRK1A
SCHEMBL19268818 0.74 APP (0.51) RIPK2RIPK3ALDH1A1HSD17B10DYRK1A
SCHEMBL8613240 0.72 NPC1 (0.46) KCNH2ALDH1A1HSD17B10
SCHEMBL16532869 0.72 PDGFRB (0.59) KCNH2ALDH1A1HSD17B10ALKCYP2E1
SCHEMBL1852870 0.71 FFAR1 (0.48) RIPK2RIPK3ALDH1A1HSD17B10DYRK1A
SCHEMBL13394464 0.71 DYRK1A (0.51) RIPK2RIPK3ALDH1A1HSD17B10DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0222970-B1 SULPHOALKYLATION PROCESS Agfa-Gevaert AG (DE) 1990-10-24 EP disclosed
US-4883880-A Process for the preparation of sulfoalkyl quaternary salts and for the production of alkane sultones AGFA-GEVAERT AKTIENGESSELLSCHAFT (DE) 1989-11-28 US disclosed
EP-0222970-A1 Sulphoalkylation process Agfa-Gevaert AG (DE) 1987-05-27 EP disclosed
US-4539408-A Process for the preparation of sulphoalkyl quaternary salts AGFA-GEVAERT AKTIENGESELLSCHAFT (DE) 1985-09-03 US disclosed
US-4504668-A Process for the preparation of N-sulfoalkyl quaternary salts of nitrogen heterocyclics AGFA-GEVAERT AKTIENGESELLSCHAFT (DE) 1985-03-12 US disclosed
EP-0064667-B1 PROCESS FOR THE PREPARATION OF SULFOALKYL QUATERNARY SALTS Agfa-Gevaert AG (DE) 1984-11-28 EP disclosed
EP-0055428-B1 BIS-(3-SULFOPROPYL)ETHERS, PROCESS FOR THEIR PREPARATION AND THEIR USE AS ALKYLATING AGENTS FOR ORGANIC BASES Agfa-Gevaert AG (DE) 1984-03-14 EP disclosed
EP-0034279-B1 SULFOALKYLATING AGENTS, PROCESS FOR THEIR PREPARATION AND THEIR USE IN THE MANUFACTURE OF QUANTERNARY SULFOALKYL SALTS Agfa-Gevaert AG (DE) 1983-06-22 EP disclosed
EP-0064667-A1 Process for the preparation of sulfoalkyl quaternary salts Agfa-Gevaert AG (DE) 1982-11-17 EP disclosed
EP-0055428-A1 Bis-(3-sulfopropyl)ethers, process for their preparation and their use as alkylating agents for organic bases Agfa-Gevaert AG (DE) 1982-07-07 EP disclosed
US-4308390-A Process for the production of sulphoalkyl quaternary salts AGFA-GEVAERT AKTIENGESELLSCHAFT (DE) 1981-12-29 US disclosed
EP-0034279-A2 Sulfoalkylating agents, process for their preparation and their use in the manufacture of quanternary sulfoalkyl salts Agfa-Gevaert AG (DE) 1981-08-26 EP disclosed