SCHEMBL10356814

SCHEMBL10356814

Cc1ccc(NCCN(C)C)nn1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.50
HRH3 Q9Y5N1 1/20 0.46
DNM2 P50570 11/20 0.42
NCF1 P14598 1/20 0.42
HRH4 Q9H3N8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1110422 0.80 CYP2C19 (0.49) CYP2C19HRH3DNM2HRH4
SCHEMBL1318627 0.80 CYP2C19 (0.49) CYP2C19HRH3DNM2HRH4L3MBTL1
SCHEMBL1752801 0.77 SYK (0.41)
SCHEMBL20037454 0.77 IL1B (0.45) CYP2C19
SCHEMBL1110459 0.75 CYP2C19 (0.47) CYP2C19HRH3DNM2NCF1HRH4
SCHEMBL15382053 0.74 HCAR3 (0.46) CYP2C19NCF1
SCHEMBL8046837 0.74 HRH3 (0.45) HRH3
SCHEMBL12895618 0.74 HCAR3 (0.39)
SCHEMBL23768365 0.73 SOAT1 (0.49) DNM2
SCHEMBL6027125 0.73 CYP2C19 (0.57) CYP2C19HRH3DNM2NCF1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121600-B1 SUBSTITUTED ARYLSULPHONYLGLYCINES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS BOEHRINGER INGELHEIM INT (DE) 2012-07-18 EP disclosed