Indole

Indole

SCHEMBL10367462

CC1CN(c2ccccc2)CC(Cl)N1.c1ccc2[nH]ccc2c1

nearest known ligand 0.45

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
ITGB2 P05107 1/20 0.45
ICAM1 P05362 1/20 0.45
ITGAL P20701 1/20 0.45
CA4 P22748 1/20 0.45
CA6 P23280 1/20 0.45
AHR P35869 1/20 0.45
ADK P55263 1/20 0.45
GHSR Q92847 6/20 0.36
BPTF Q12830 1/20 0.36
SLC6A4 P31645 3/20 0.34
SLC6A2 P23975 2/20 0.34
SLC6A3 Q01959 2/20 0.34
MAPK14 Q16539 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
HTR2C P28335 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Indole SCHEMBL10364968 0.79 TRPA1 (0.40) TRPA1CA1CA2ITGB2ICAM1
SCHEMBL12663143 0.74 BPTF (0.53) GHSRBPTFALDH1A1HTR2CKHK
SCHEMBL8342001 0.74 BPTF (0.53) BPTFSLC6A4HTR2CKCNH2
SCHEMBL800968 0.74 BPTF (0.53) GHSRBPTFALDH1A1HTR2CKHK
Indole SCHEMBL27977912 0.69 TRPA1 (0.59) TRPA1CA1CA2ITGB2ICAM1
Indole SCHEMBL30877947 0.69 AHR (0.94) TRPA1CA1CA2ITGB2ICAM1
Indole SCHEMBL2945202 0.69 AHR (0.94) TRPA1CA1CA2ITGB2ICAM1
Indole SCHEMBL27957692 0.67 AHR (0.90) TRPA1CA1CA2ITGB2ICAM1
Indole SCHEMBL6386255 0.67 AHR (0.90) TRPA1CA1CA2ITGB2ICAM1
Indole SCHEMBL698 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0200322-B1 HETEROCYCLIC COMPOUNDS H. LUNDBECK A/S (DK) 1990-02-28 EP disclosed
US-4710500-A 1-(4'-fluorophenyl)-3,5-substituted indoles useful in the treatment of psychic disorders and pharmaceutical compositions thereof H. LUNDBECK A/S (DK) 1987-12-01 US disclosed
EP-0200322-A1 Heterocyclic compounds H. LUNDBECK A/S (DK) 1986-11-05 EP disclosed