SCHEMBL10375772

SCHEMBL10375772

CN(C)c1cc(N)nc(N(C)C)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.43
CYP1A2 P05177 1/20 0.43
THRB P10828 1/20 0.43
BLM P54132 1/20 0.43
CREBBP Q92793 1/20 0.43
HSD17B10 Q99714 1/20 0.43
NUDT1 P36639 1/20 0.42
MAPT P10636 4/20 0.38
APAF1 O14727 4/20 0.38
NSD2 O96028 3/20 0.38
SAE1 Q9UBE0 3/20 0.38
UBA2 Q9UBT2 3/20 0.38
SENP8 Q96LD8 3/20 0.38
SENP7 Q9BQF6 3/20 0.38
SENP6 Q9GZR1 3/20 0.38
CASP3 P42574 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
KDM4E B2RXH2 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10377966 0.85 LMNA (0.53) LMNACYP1A2THRBBLMCREBBP
SCHEMBL4265950 0.83 LMNA (0.56) LMNACYP1A2THRBBLMCREBBP
SCHEMBL11481158 0.77 NOS3 (0.48) LMNACYP1A2THRBBLMCREBBP
SCHEMBL4256097 0.77 NUDT1 (0.42) NUDT1KMT2AMEN1TSHRNOS3
SCHEMBL2467611 0.76 LMNA (0.42) LMNACYP1A2THRBBLMCREBBP
SCHEMBL11398865 0.76 LMNA (0.42) LMNACYP1A2THRBBLMCREBBP
SCHEMBL13780086 0.74 MEN1 (0.59) LMNACYP1A2THRBBLMCREBBP
SCHEMBL9270907 0.73 LMNA (0.43) LMNACYP1A2THRBBLMCREBBP
SCHEMBL2789514 0.73 KMT2A (0.47) LMNACYP1A2THRBBLMCREBBP
SCHEMBL9380659 0.72 LMNA (0.44) LMNACYP1A2THRBBLMCREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-59200253-A None JP disclosed
EP-0189045-B1 PYRIDOPYRIMIDINES, DIFFERENT PROCESSES FOR THEIR PREPARATION AS WELL AS THEIR USE AS MEDICAMENTS BAYER AG (DE) 1990-02-14 EP disclosed
US-4621082-A Pyridopyrimidines, pharmaceutical compositions and use BAYER AKTIENGESELLSCHAFT (DE) 1986-11-04 US disclosed
EP-0189045-A2 Pyridopyrimidines, different processes for their preparation as well as their use as medicaments BAYER AG (DE) 1986-07-30 EP disclosed
JP-S59200253-A POSITIVE ELECTROSTATIC CHEARGEABLE TONER FOR TWO- COMPONENT DEVELOPER FUJITSU LTD 1984-11-13 JP disclosed
US-4331805-A OPTICAL BRIGHTENERS CIBA-GEIGY CORPORATION (US) 1982-05-25 US disclosed
US-4236003-A OPTICAL BRIGHTENERS CIBA-GEIGY CORPORATION (US) 1980-11-25 US disclosed
US-4157443-A OPTICAL BRIGHTENERS CIBA-GEIGY CORPORATION (US) 1979-06-05 US disclosed