SCHEMBL10378306

SCHEMBL10378306

CC(C)C([C]=O)NC(=O)C1CCCN1CC(Cc1ccccc1)NC(=O)C(CC(N)=O)NC(=O)C(CCC(N)=O)NC(=O)C(N)CO

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA2B P29275 1/20 0.41
ADORA1 P30542 1/20 0.41
BACE1 P56817 5/20 0.40
NMUR2 Q9GZQ4 2/20 0.39
NMUR1 Q9HB89 2/20 0.39
F2 P00734 1/20 0.39
REN P00797 1/20 0.38
OPRD1 P41143 2/20 0.38
HRH1 P35367 2/20 0.38
CALCRL Q16602 1/20 0.38
OPRM1 P35372 1/20 0.37
OPRK1 P41145 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7326543 0.93 NMUR2 (0.41) ADORA3ADORA2AADORA2BADORA1NMUR2
SCHEMBL10378303 0.91 HRH1 (0.41) ADORA3ADORA2AADORA2BADORA1NMUR2
SCHEMBL10376958 0.88 F2 (0.43) ADORA3ADORA2AADORA2BADORA1F2
SCHEMBL7329810 0.77 CTRB1 (0.43) F2
SCHEMBL7320110 0.77 CTSD (0.50) ADORA3ADORA2AADORA2BADORA1BACE1
SCHEMBL7330209 0.76 BACE1 (0.51) BACE1REN
SCHEMBL7328124 0.76 BACE1 (0.51) BACE1REN
SCHEMBL7328119 0.76 BACE1 (0.51) BACE1REN
SCHEMBL7331125 0.74 CTSD (0.43) NMUR2NMUR1F2CALCRL
SCHEMBL10376833 0.74 NMUR2 (0.51) NMUR2NMUR1F2OPRD1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1990000399-A1 RETROVIRAL PROTEASE BINDING PEPTIDES SMITHKLINE BECKMAN CORPORATION (US) 1990-01-25 WO claimed
WO-1990000399-A1 RETROVIRAL PROTEASE BINDING PEPTIDES SMITHKLINE BECKMAN CORPORATION (US) 1990-01-25 WO disclosed