SCHEMBL10396604

SCHEMBL10396604

CN(Cc1ccc2ccccc2c1)C(=O)n1ccnc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.49
MGLL Q99685 1/20 0.49
CYP19A1 P11511 2/20 0.49
CYP2D6 P10635 1/20 0.42
TBXAS1 P24557 2/20 0.41
PYCR1 P32322 1/20 0.40
PDK1 Q15118 1/20 0.40
PDK2 Q15119 1/20 0.40
PDK3 Q15120 1/20 0.40
PDK4 Q16654 1/20 0.40
CYP11B1 P15538 2/20 0.40
CYP11B2 P19099 2/20 0.40
ACHE P22303 1/20 0.40
ALDH1A1 P00352 1/20 0.39
GBA1 P04062 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
CYP26A1 O43174 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5648204 0.84 CYP1A2 (0.51) CYP19A1CYP2D6
SCHEMBL19691848 0.79 ALDH1A1 (0.50) CYP19A1CYP2D6CYP11B1CYP11B2ALDH1A1
SCHEMBL10543520 0.74 POLB (0.43) CYP19A1CYP2D6CYP11B1CYP11B2CYP26A1
SCHEMBL23972322 0.73 SLC6A2 (0.55) TRPV1MGLLPYCR1PDK1PDK2
SCHEMBL26027596 0.73 TRPV1 (0.51) TRPV1MGLLPYCR1ACHESLC6A2
SCHEMBL15435863 0.72 CYP19A1 (0.49) MGLLCYP19A1CYP2D6TBXAS1CYP11B1
SCHEMBL10545302 0.72 PPARG (0.44) TBXAS1CYP26A1
SCHEMBL10397484 0.72 PYCR1 (0.50) TRPV1MGLLPYCR1PDK1ACHE
SCHEMBL20111609 0.72 LIPE (0.48) CYP2D6ALDH1A1
SCHEMBL1171099 0.71 AHR (0.42) TBXAS1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4840961-A FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 1989-06-20 US claimed
US-4952595-A FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 1990-08-28 US disclosed
US-4840961-A FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 1989-06-20 US disclosed
EP-0198382-A2 Heterocyclic amide derivatives BAYER AG (DE) 1986-10-22 EP disclosed