SCHEMBL10399189

SCHEMBL10399189

CCOC(=O)/C=C/C=C(c1cccc(C(F)(F)F)c1)c1cccc(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.47
ALDH1A1 P00352 2/20 0.46
POLB P06746 1/20 0.46
NPSR1 Q6W5P4 1/20 0.45
MAPT P10636 2/20 0.44
TAS1R3 Q7RTX0 1/20 0.43
TAS1R1 Q7RTX1 1/20 0.43
MAOB P27338 1/20 0.43
F2 P00734 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
HTT P42858 2/20 0.42
GAA P10253 1/20 0.41
MEN1 O00255 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10399109 1.00 CES2 (0.47) CES2ALDH1A1POLBNPSR1MAPT
SCHEMBL10399108 1.00 CES2 (0.47) CES2ALDH1A1POLBNPSR1MAPT
SCHEMBL3938552 0.85 MAPT (0.45) ALDH1A1POLBNPSR1MAPTMAOB
SCHEMBL3938554 0.85 MAPT (0.45) ALDH1A1POLBNPSR1MAPTMAOB
SCHEMBL3269421 0.84 NPSR1 (0.52) CES2ALDH1A1POLBNPSR1MAPT
SCHEMBL24951715 0.83 ALDH1A1 (0.59) CES2ALDH1A1POLBNPSR1MAPT
SCHEMBL10397671 0.83 LMNA (0.49) CES2ALDH1A1POLBNPSR1MAPT
SCHEMBL10397670 0.83 LMNA (0.49) CES2ALDH1A1POLBNPSR1MAPT
SCHEMBL28630576 0.83 ALDH1A1 (0.59) CES2ALDH1A1POLBNPSR1MAPT
SCHEMBL10398662 0.81 PTAFR (0.45) ALDH1A1MAPTMAOBHTTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4975438-A ANTICOAGULANT HOFFMANN-LA ROCHE INC. (US) 1990-12-04 US disclosed
US-4788206-A CARDIOVASCULAR DISORDERS, PLATELETS HOFFMANN-LA ROCHE INC. (US) 1988-11-29 US disclosed