SCHEMBL10401282

SCHEMBL10401282

COc1cc2nc(C#N)sc2cc1OC

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
STING1 Q86WV6 1/20 0.44
ALOX15 P16050 1/20 0.43
ATM Q13315 1/20 0.43
PGK1 P00558 5/20 0.42
NSD2 O96028 5/20 0.40
QPCT Q16769 1/20 0.40
NQO2 P16083 1/20 0.39
KDM4E B2RXH2 1/20 0.38
IKBKE Q14164 1/20 0.37
USP8 P40818 1/20 0.36
USP7 Q93009 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21663984 0.89 ALOX15 (0.43) STING1ALOX15ATMPGK1NSD2
SCHEMBL935080 0.87 PGK1 (0.47) ALOX15ATMPGK1
SCHEMBL21688901 0.87 ALOX15 (0.39) STING1ALOX15ATMPGK1NSD2
SCHEMBL12312875 0.87 ILK (0.47) ALOX15ATM
SCHEMBL12312873 0.87 PGK1 (0.47) STING1ALOX15ATMPGK1
SCHEMBL935523 0.84 CTSS (0.40) ALOX15ATM
SCHEMBL9796864 0.81 PSMB8 (0.44)
SCHEMBL5857526 0.77 NPC1 (0.54) ALOX15KDM4E
SCHEMBL906609 0.77 CYP1A2 (0.59)
SCHEMBL12908847 0.77 GAA (0.57) NQO2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4929636-A Positive inotrophic benzothiazole and benzothiophene compositions and method of use therefor AKZO N.V. (NL) 1990-05-29 US disclosed
EP-0158380-B1 BENZOTHIAZOLE AND BENZOTHIOPHENE DERIVATIVES AKZO N.V. (NL) 1989-01-11 EP disclosed
US-4665206-A Benzothiophene derivatives AKZO N.V. (NL) 1987-05-12 US disclosed
EP-0158380-A1 Benzothiazole and benzothiophene derivatives AKZO N.V. (NL) 1985-10-16 EP disclosed