SCHEMBL10409233

SCHEMBL10409233

Nc1cccc(C(=O)N2CC3CN(Cc4ccccc4)CC(C2)C3=O)c1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.54
MAPK1 P28482 2/20 0.54
MEN1 O00255 1/20 0.54
LMNA P02545 1/20 0.54
KMT2A Q03164 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
HSD11B1 P28845 1/20 0.47
ALDH1A1 P00352 2/20 0.46
KDM4E B2RXH2 1/20 0.46
ADRB2 P07550 1/20 0.45
CYP2D6 P10635 3/20 0.45
DRD2 P14416 1/20 0.44
DRD4 P21917 1/20 0.44
NPC1 O15118 1/20 0.44
MGLL Q99685 1/20 0.44
RECQL P46063 1/20 0.43
CHRM2 P08172 1/20 0.43
CHRM3 P20309 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10409232 0.87 MAPK1 (0.55) TSHRMAPK1MEN1LMNAKMT2A
SCHEMBL10410773 0.80 KDM4E (0.50) ALDH1A1KDM4EDRD2DRD4CHRM2
SCHEMBL6609510 0.78 S1PR5 (0.53) TSHRMEN1LMNAKMT2ASMN1; SMN2
SCHEMBL2962712 0.76 FUCA1 (0.58) TSHR
SCHEMBL10409277 0.75 HTT (0.57) LMNAKMT2ASMN1; SMN2ALDH1A1KDM4E
Ambasilide SCHEMBL427931 0.74 HSD11B1 (0.53) TSHRMAPK1MEN1LMNAKMT2A
Ambasilide SCHEMBL246531 0.74 HSD11B1 (0.53) TSHRMAPK1MEN1LMNAKMT2A
SCHEMBL17953046 0.74 KDM4E (0.61) TSHRMAPK1MEN1LMNAKMT2A
SCHEMBL22702112 0.73 CA12 (0.54) LMNAL3MBTL1ALDH1A1KDM4ENPC1
SCHEMBL29804524 0.73 CA12 (0.54) LMNAL3MBTL1ALDH1A1KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4959373-A Bispidine derivatives as class III antiarrhythmic agents BASF AKTIENGESELLSCHAFT (DE) 1990-09-25 US disclosed