SCHEMBL10412436

SCHEMBL10412436

CON=C(C(C)=Cc1ccc(OC(F)(F)F)cc1)C(C)n1cncn1

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 3/20 0.33
KMT2A Q03164 3/20 0.33
MAPT P10636 1/20 0.33
POLB P06746 1/20 0.32
HSP90AA1 P07900 1/20 0.32
CYP3A4 P08684 1/20 0.32
MEN1 O00255 2/20 0.31
TDP1 Q9NUW8 1/20 0.31
CYP19A1 P11511 1/20 0.31
GRM7 Q14831 1/20 0.31
LMNA P02545 1/20 0.31
KDM4E B2RXH2 1/20 0.30
PDE2A O00408 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10414102 0.74 SLC6A4 (0.36) KMT2APOLBHSP90AA1MEN1CYP19A1
SCHEMBL9362870 0.73 APP (0.43) CYP3A4LMNA
SCHEMBL9362865 0.73 APP (0.43) CYP3A4LMNA
SCHEMBL9467685 0.71 POLB (0.38) KMT2AMAPTPOLBHSP90AA1CYP3A4
SCHEMBL9467692 0.71 POLB (0.38) KMT2AMAPTPOLBHSP90AA1CYP3A4
SCHEMBL10568532 0.70 HSP90AA1 (0.47) KMT2AHSP90AA1CYP3A4GRM7LMNA
SCHEMBL10360787 0.66 HSP90AA1 (0.42) KMT2APOLBHSP90AA1CYP3A4MEN1
SCHEMBL9366526 0.66 ALDH1A1 (0.42) KMT2AMAPTCYP3A4MEN1CYP19A1
SCHEMBL10565684 0.66 CYP19A1 (0.40) KMT2APOLBHSP90AA1CYP3A4MEN1
SCHEMBL10565622 0.66 PDE2A (0.44) KMT2APOLBHSP90AA1CYP3A4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4962118-A ACTIVE AGAINST ASPERGILLUS, CHAETOMIUM, PENICILLUM; WHEAT, BARLEY BAYER AKTIENGESELLSCHAFT (DE) 1990-10-09 US claimed