SCHEMBL10416359

SCHEMBL10416359

COC(=O)N1CCNC(CO)C1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.42
CHRNA4 P43681 3/20 0.42
CHRNA3 P32297 2/20 0.42
CHRNB4 P30926 1/20 0.42
REN P00797 4/20 0.39
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36
CA4 P22748 2/20 0.36
CA9 Q16790 2/20 0.36
TSHR P16473 1/20 0.35
SCN9A Q15858 4/20 0.35
CHRNB3 Q05901 1/20 0.34
CHRNA6 Q15825 1/20 0.34
BIRC2 Q13490 1/20 0.33
CYP2D6 P10635 1/20 0.33
ITGB2 P05107 1/20 0.32
ICAM1 P05362 1/20 0.32
ITGAL P20701 1/20 0.32
TPSAB1 Q15661 1/20 0.32
TPSD1 Q9BZJ3 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28750702 0.85 ALDH1A1 (0.43) RENTSHR
SCHEMBL29270907 0.85 ALDH1A1 (0.43) RENTSHR
SCHEMBL26741797 0.85 REN (0.40) CHRNB2CHRNA4CHRNA3RENCA1
SCHEMBL5190958 0.83 CHRNB2 (0.39) CHRNB2CHRNA4CHRNA3CHRNB4REN
SCHEMBL336866 0.83 NR1H2 (0.50) REN
SCHEMBL1462710 0.83 NR1H2 (0.50) REN
SCHEMBL994990 0.83 NR1H2 (0.50) REN
SCHEMBL15360065 0.82 CHRNB2 (0.47) CHRNB2CHRNA4CHRNA3CHRNB4REN
SCHEMBL4332763 0.82 CHRNB2 (0.47) CHRNB2CHRNA4CHRNA3CHRNB4REN
SCHEMBL15360066 0.82 CHRNB2 (0.47) CHRNB2CHRNA4CHRNA3CHRNB4REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4943578-A ANALGESICS; CEREBRAL ANTIISCHEMIC AGENTS GLAXO GROUP LIMITED (GB) 1990-07-24 US disclosed
EP-0343900-A2 Piperazine compounds GLAXO GROUP LIMITED (GB) 1989-11-29 EP disclosed