SCHEMBL5190958

SCHEMBL5190958

COC(=O)N1CCNC(CC(N)=O)C1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.39
CHRNA4 P43681 2/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
CA1 P00915 4/20 0.34
CA2 P00918 4/20 0.34
CA4 P22748 4/20 0.34
CA9 Q16790 4/20 0.34
PARP1 P09874 1/20 0.34
TSHR P16473 1/20 0.33
REN P00797 1/20 0.32
BIRC2 Q13490 1/20 0.31
PDE4B Q07343 3/20 0.31
PDE4A P27815 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
CYP2D6 P10635 1/20 0.31
CCR3 P51677 1/20 0.31
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31436244 0.84 NR1H2 (0.40) PDE4B
SCHEMBL31436240 0.84 NR1H2 (0.40) PDE4B
SCHEMBL10416359 0.83 CHRNB2 (0.42) CHRNB2CHRNA4CHRNB4CHRNA3CA1
SCHEMBL7063658 0.81 NPY2R (0.41) CHRNB2CHRNA4CHRNB4CHRNA3CYP2D6
SCHEMBL27470540 0.78 OPRM1 (0.40) CHRNB2CHRNA4CHRNB4CHRNA3BIRC2
SCHEMBL7670875 0.78 OPRM1 (0.40) CHRNB2CHRNA4CHRNB4CHRNA3BIRC2
SCHEMBL17560422 0.76 CHRNB2 (0.42) CHRNB2CHRNA4CHRNB4CHRNA3TSHR
SCHEMBL24721279 0.76 BIRC2 (0.32) PARP1BIRC2
SCHEMBL2918458 0.76 BIRC2 (0.32) PARP1BIRC2
SCHEMBL5193199 0.75 MAPT (0.55) TSHRCYP2D6CCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP claimed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP claimed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO claimed