SCHEMBL10418367

SCHEMBL10418367

COc1ccc2c(N(C)c3ccc(O)cc3)cccc2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
CYP2A6 P11509 1/20 0.41
MCL1 Q07820 1/20 0.41
MTNR1A P48039 5/20 0.40
MTNR1B P49286 4/20 0.40
HTR2A P28223 1/20 0.38
MEN1 O00255 1/20 0.38
CASP3 P42574 1/20 0.38
KMT2A Q03164 1/20 0.38
SENP8 Q96LD8 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
SENP6 Q9GZR1 1/20 0.38
C5AR1 P21730 1/20 0.38
LTA4H P09960 1/20 0.38
ESR2 Q92731 1/20 0.38
HSP90AA1 P07900 1/20 0.37
PDK1 Q15118 1/20 0.37
PDK2 Q15119 1/20 0.37
PDK3 Q15120 1/20 0.37
PDK4 Q16654 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12048740 0.79 EGFR (0.51) CASP3KMT2A
SCHEMBL12060551 0.79 SIGMAR1 (0.53) CYP1A2MCL1MEN1KMT2A
SCHEMBL4600762 0.79 CYP1A2 (0.52) CYP1A2CYP2A6MCL1MTNR1AMTNR1B
SCHEMBL9702074 0.77 CYP1A1 (0.46) CYP1A2CYP2A6MTNR1AMTNR1BMEN1
SCHEMBL9290859 0.75 XDH (0.46) CYP1A2CYP2A6MEN1KMT2ALTA4H
Mequinol SCHEMBL8923068 0.74 MCL1 (0.58) CYP1A2CYP2A6MCL1MEN1KMT2A
SCHEMBL17602315 0.74 MTNR1A (0.62) MTNR1AMTNR1BMEN1KMT2A
SCHEMBL12048742 0.74 DHFR (0.45) CYP1A2CYP2A6MTNR1AMTNR1BHTR2A
SCHEMBL17602128 0.73 ESR2 (0.61) CASP3SENP8SENP7SENP6LTA4H
SCHEMBL9163161 0.72 CYP1A2 (0.45) CYP1A2CYP2A6MTNR1AMTNR1BMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4910208-A Skin disorders, antiinflammatory agent E. R. SQUIBB & SONS, INC. (US) 1990-03-20 US claimed