SCHEMBL10418486

SCHEMBL10418486

c1ccc(N(c2ccccc2)c2cc[nH]n2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.40
ALDH1A1 P00352 4/20 0.38
MAPT P10636 3/20 0.38
TDP1 Q9NUW8 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
KDM4E B2RXH2 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
TAAR1 Q96RJ0 2/20 0.33
MEN1 O00255 1/20 0.32
CRHBP P24387 1/20 0.32
KMT2A Q03164 1/20 0.32
ATM Q13315 1/20 0.32
CRHR2 Q13324 1/20 0.32
TLR9 Q9NR96 1/20 0.32
KCNA3 P22001 1/20 0.32
EGFR P00533 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4690140 0.78 NPSR1 (0.32) POLBALDH1A1MAPTTDP1L3MBTL1
SCHEMBL17674048 0.78 DHFR (0.42) TAAR1MEN1KMT2AEGFRCSF1R
SCHEMBL1667246 0.74 ALDH1A1 (0.38) POLBALDH1A1ALOX15
SCHEMBL17049294 0.74 POLB (0.32) POLB
SCHEMBL4458935 0.74 NPSR1 (0.47) POLBALDH1A1MAPTTDP1L3MBTL1
SCHEMBL6905225 0.71 KMT2A (0.46) POLBALDH1A1TDP1L3MBTL1MEN1
SCHEMBL398536 0.71 NPSR1 (0.44) POLBALDH1A1TDP1L3MBTL1MEN1
SCHEMBL11342835 0.71 ESR1 (0.35) ALDH1A1MAPTL3MBTL1KDM4ECYP1A2
SCHEMBL12668168 0.70 ALDH1A1 (0.44) POLBALDH1A1MAPTTDP1L3MBTL1
SCHEMBL4268460 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0178035-B1 ANTI-INFLAMMATORY 1,N-DIARYLPYRAZOL-3-AMINES, COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION FISONS plc (GB) 1990-01-03 EP claimed