SCHEMBL10426328

SCHEMBL10426328

C=Cc1ccnc(C)c1C=C

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDXK O00764 1/20 0.35
CYP2A6 P11509 1/20 0.34
HDAC8 Q9BY41 1/20 0.32
CCR1 P32246 2/20 0.30
CCR5 P51681 2/20 0.30
CCR8 P51685 2/20 0.30
UHRF1 Q96T88 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19443439 0.85 CCR1 (0.39) CYP2A6CCR1CCR5CCR8
SCHEMBL21340202 0.84 PDXK (0.32) PDXKCYP2A6
SCHEMBL26462240 0.82
SCHEMBL4944670 0.82 CCR1 (0.34) PDXKCYP2A6HDAC8CCR1CCR5
SCHEMBL29673267 0.82 CCR1 (0.34) PDXKCYP2A6HDAC8CCR1CCR5
SCHEMBL11830120 0.79 NOS2 (0.40) PDXKCYP2A6
SCHEMBL15417589 0.79 CCR1 (0.39) PDXKCYP2A6HDAC8CCR1CCR5
SCHEMBL9467052 0.77 CCR1 (0.30) CCR1CCR5CCR8
SCHEMBL1522103 0.77 PDXK (0.35) PDXKCYP2A6HDAC8CCR1CCR5
SCHEMBL25777478 0.76 ALDH1A1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021225912-A1 TREATMENT OF RESPIRATORY DISEASES WITH AMINO ACID COMPOUNDS PLIANT THERAPEUTICS, INC. (US) 2021-11-11 WO disclosed
US-4943482-A ADDITION COPOLYMER WITH SILVER OR PALLADIUM COATING RHONE-POULENC CHIMIE (FR) 1990-07-24 US disclosed
EP-0311476-A1 Metallized particles of crosslinked functional polymers, their preparation and their use in producing electroconductive materials RHONE-POULENC CHIMIE (FR) 1989-04-12 EP disclosed
EP-0103538-A2 Copolymers of vinylpyridine, process for their preparation and their use as sulphonate reagents CIBA-GEIGY AG (CH) 1984-03-21 EP disclosed