SCHEMBL10429339

SCHEMBL10429339

O=c1[nH]nnc2c(-c3ccc(Br)cc3)nsc12

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.33
POLB P06746 1/20 0.33
RAB9A P51151 1/20 0.33
ATM Q13315 1/20 0.33
KDM4E B2RXH2 1/20 0.32
PKM P14618 1/20 0.32
GRM5 P41594 1/20 0.32
GRM1 Q13255 1/20 0.32
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
TNKS O95271 3/20 0.30
TNKS2 Q9H2K2 3/20 0.30
PARP1 P09874 1/20 0.30
PARP2 Q9UGN5 1/20 0.30
PDE3B Q13370 1/20 0.30
PDE3A Q14432 1/20 0.30
CYP1A1 P04798 1/20 0.30
CYP1B1 Q16678 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10429350 0.85 KDR (0.36) ALDH1A1HPGDTNKSTNKS2PARP1
SCHEMBL10429322 0.85 ALDH1A1 (0.37) NPC1RAB9AKDM4EGRM5GRM1
SCHEMBL2121780 0.85 NPSR1 (0.40) NPC1POLBRAB9AATMKDM4E
Hydrochloric Acid SCHEMBL10429329 0.84 KDR (0.35) ALDH1A1HPGDPDE3BPDE3A
SCHEMBL10429361 0.83 MAOB (0.36) NPC1POLBRAB9AKDM4EPKM
SCHEMBL10429313 0.83 NOTUM (0.38) POLBKDM4EALDH1A1HPGDKMT2A
SCHEMBL10429367 0.82 HPGD (0.47) NPC1POLBRAB9AKDM4EALDH1A1
SCHEMBL10429337 0.81 XDH (0.40) PKMALDH1A1HPGDMEN1KMT2A
SCHEMBL10429340 0.78 NOTUM (0.39) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL10429304 0.78 SMN1; SMN2 (0.43) NPC1POLBRAB9AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0274654-A2 1,2,3-Triazin-4(3H)-one derivatives, process for their preparation and medicaments containing them F. HOFFMANN-LA ROCHE AG (CH) 1988-07-20 EP claimed
US-4920119-A XANTHINE OXIDASE INHIBITORS; CONTROL OR PREVENTION OF GOUT OR ISCHEMIA HOFFMANN-LA ROCHE INC. (US) 1990-04-24 US disclosed
EP-0274654-A2 1,2,3-Triazin-4(3H)-one derivatives, process for their preparation and medicaments containing them F. HOFFMANN-LA ROCHE AG (CH) 1988-07-20 EP disclosed