SCHEMBL10429340

SCHEMBL10429340

O=c1[nH]nnc2c(-c3ccc4ccccc4c3)nsc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.39
CA12 O43570 1/20 0.37
MAOB P27338 1/20 0.37
GSTP1 P09211 1/20 0.37
MAPK8 P45983 1/20 0.37
MAPK9 P45984 1/20 0.37
MAPK10 P53779 1/20 0.37
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
ALDH1A1 P00352 4/20 0.35
CYP1A2 P05177 2/20 0.35
HPGD P15428 2/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
NOS1 P29475 1/20 0.35
ALPL P05186 1/20 0.34
PDGFRB P09619 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
HTR2B P41595 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10429321 0.79 ADORA3 (0.39) NOTUMALDH1A1CYP1A2HPGDCYP2C9
SCHEMBL10429361 0.79 MAOB (0.36) MAOBALDH1A1CYP1A2HPGDCYP2C9
SCHEMBL10429350 0.78 KDR (0.36) ALDH1A1HPGDALPLPDGFRB
SCHEMBL10429322 0.78 ALDH1A1 (0.37) NOTUMCA12ADORA2AADORA1ALDH1A1
SCHEMBL10429367 0.77 HPGD (0.47) NOTUMALDH1A1CYP1A2HPGDCYP2C9
SCHEMBL10429323 0.76 MAOB (0.40) NOTUMMAOBADORA2AADORA1
SCHEMBL10429313 0.76 NOTUM (0.38) NOTUMCA12ALDH1A1HPGDALPL
SCHEMBL10429364 0.75 NOTUM (0.33) NOTUMALDH1A1HPGD
SCHEMBL7162696 0.74 PDE4A (0.38) MAOBADORA2AADORA1ALDH1A1HPGD
SCHEMBL10429334 0.73 NOTUM (0.40) NOTUMSMN1; SMN2NPC1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0274654-A2 1,2,3-Triazin-4(3H)-one derivatives, process for their preparation and medicaments containing them F. HOFFMANN-LA ROCHE AG (CH) 1988-07-20 EP claimed
US-4920119-A XANTHINE OXIDASE INHIBITORS; CONTROL OR PREVENTION OF GOUT OR ISCHEMIA HOFFMANN-LA ROCHE INC. (US) 1990-04-24 US disclosed