SCHEMBL10429367

SCHEMBL10429367

COc1ccc(-c2nsc3c(=O)[nH]nnc23)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 6/20 0.47
ALDH1A1 P00352 6/20 0.47
KDM4E B2RXH2 6/20 0.44
RAB9A P51151 5/20 0.44
SMN1; SMN2 Q16637 5/20 0.44
MAPT P10636 5/20 0.44
NPC1 O15118 3/20 0.44
TP53 P04637 2/20 0.44
RXFP1 Q9HBX9 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.39
LMNA P02545 1/20 0.38
CCNE2 O96020 2/20 0.38
CDK4 P11802 2/20 0.38
CCND1 P24385 2/20 0.38
CCNE1 P24864 2/20 0.38
CDK2 P24941 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10429305 0.85 NOTUM (0.42) HPGDALDH1A1SMN1; SMN2MAPTLMNA
SCHEMBL10429322 0.82 ALDH1A1 (0.37) HPGDALDH1A1KDM4ERAB9ASMN1; SMN2
SCHEMBL2121780 0.81 NPSR1 (0.40) HPGDALDH1A1KDM4ERAB9ASMN1; SMN2
Hydrochloric Acid SCHEMBL10429329 0.81 KDR (0.35) HPGDALDH1A1
SCHEMBL7165524 0.80 GRM5 (0.41) HPGDALDH1A1KDM4ERAB9ASMN1; SMN2
SCHEMBL7162696 0.80 PDE4A (0.38) HPGDALDH1A1MAPTTP53LMNA
SCHEMBL7166176 0.79 GSTP1 (0.44) HPGDRAB9ASMN1; SMN2NPC1L3MBTL1
SCHEMBL7162474 0.78 CTSS (0.37) HPGDALDH1A1GSK3B
SCHEMBL7165222 0.78 F11 (0.40) ALDH1A1KDM4E
SCHEMBL10429340 0.77 NOTUM (0.39) HPGDALDH1A1KDM4ERAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0274654-A2 1,2,3-Triazin-4(3H)-one derivatives, process for their preparation and medicaments containing them F. HOFFMANN-LA ROCHE AG (CH) 1988-07-20 EP claimed
US-4920119-A XANTHINE OXIDASE INHIBITORS; CONTROL OR PREVENTION OF GOUT OR ISCHEMIA HOFFMANN-LA ROCHE INC. (US) 1990-04-24 US disclosed
EP-0274654-A2 1,2,3-Triazin-4(3H)-one derivatives, process for their preparation and medicaments containing them F. HOFFMANN-LA ROCHE AG (CH) 1988-07-20 EP disclosed