SCHEMBL10429391

SCHEMBL10429391

Cc1nc2ccc(-c3ccccn3)c(N)c2[nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.42
PKM P14618 5/20 0.42
RAB9A P51151 5/20 0.42
KDM4E B2RXH2 5/20 0.42
METAP2 P50579 4/20 0.42
CBFB Q13951 4/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
METAP1 P53582 3/20 0.42
L3MBTL1 Q9Y468 3/20 0.42
HPGD P15428 3/20 0.42
LMNA P02545 2/20 0.42
TP53 P04637 2/20 0.42
GAA P10253 2/20 0.42
PI4KA P42356 1/20 0.42
PI4K2B Q8TCG2 1/20 0.42
PI4K2A Q9BTU6 1/20 0.42
PI4KB Q9UBF8 1/20 0.42
MAPT P10636 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
ALOX15 P16050 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4313385 0.82 NPC1 (0.45) NPC1PKMRAB9AKDM4EMETAP2
SCHEMBL10146529 0.70 MAPT (0.52) NPC1KDM4ESMN1; SMN2L3MBTL1LMNA
SCHEMBL28996530 0.70 POLB (0.55) NPC1PKMRAB9AKDM4EMETAP2
SCHEMBL30428608 0.70 POLB (0.55) NPC1PKMRAB9AKDM4EMETAP2
SCHEMBL16503975 0.68 SMN1; SMN2 (0.47) NPC1PKMRAB9AKDM4ECBFB
SCHEMBL28171197 0.68 TYMS (0.38) NPC1RAB9AKDM4ESMN1; SMN2L3MBTL1
SCHEMBL13383928 0.68 ALDH1A1 (0.48) NPC1PKMRAB9AKDM4ESMN1; SMN2
SCHEMBL27545882 0.68 KDM4E (0.50) NPC1PKMRAB9AKDM4ESMN1; SMN2
SCHEMBL7910798 0.67 KDM4E (0.46) NPC1PKMRAB9AKDM4ESMN1; SMN2
SCHEMBL8296009 0.66 NOS2 (0.41) NPC1RAB9AKDM4EGAAPI4KA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4956351-A INCLUSION COMPLEXESOFVIRICIDES; RHINITIS; SUSTAINED RELEASE; NONIRRITATING TO MUCOUS MEMBRANE JANSSEN PHARMACEUTICA N.V. FRAME-543 (BE) 1990-09-11 US disclosed
EP-0300526-A2 Antiviral pharmaceutical compositions containing cyclodextrins JANSSEN PHARMACEUTICA N.V. (BE) 1989-01-25 EP disclosed