SCHEMBL10437460

SCHEMBL10437460

O=c1[nH]c2ccc(Nc3ccc(O)nc3)cc2o1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.49
NOS1 P29475 1/20 0.44
JAK1 P23458 1/20 0.44
JAK3 P52333 1/20 0.44
CREBBP Q92793 1/20 0.44
MAPKAPK2 P49137 6/20 0.43
PDE3B Q13370 1/20 0.43
PDE3A Q14432 1/20 0.43
IRAK4 Q9NWZ3 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
P2RX3 P56373 1/20 0.41
POLB P06746 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
TSHR P16473 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10338403 0.77 PDE3B (0.61) SYKNOS1JAK1JAK3CREBBP
SCHEMBL10359665 0.77 SYK (0.55) SYKNOS1JAK1JAK3CREBBP
SCHEMBL21925302 0.77 SYK (0.56) SYKNOS1JAK1JAK3CREBBP
SCHEMBL10437432 0.73 SYK (0.49) SYKNOS1JAK1JAK3CREBBP
SCHEMBL10437441 0.73 SYK (0.46) SYKNOS1JAK1JAK3CREBBP
SCHEMBL14465953 0.73 FLT1 (0.58) SYKJAK1JAK3MAPKAPK2PDE3B
SCHEMBL10437477 0.72 SYK (0.48) SYKNOS1JAK1JAK3CREBBP
SCHEMBL5321701 0.72 ALOX5 (0.52) SYKPDE3BPDE3A
SCHEMBL8311380 0.71 NOS1 (0.61) SYKNOS1CREBBPPDE3BPDE3A
SCHEMBL10437451 0.71 SYK (0.50) SYKNOS1JAK1JAK3CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0360566-A2 Lipoxygenase/cyclooxygenase inhibiting benzoxazolones PFIZER INC. (US) 1990-03-28 EP disclosed