SCHEMBL10444544

SCHEMBL10444544

C=C1C[C@H]2[C@@H]3C=C(C)C4=CC(=O)CC[C@]4(C)[C@H]3CC[C@]2(C)C1=O

nearest known ligand 0.69

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 14/20 0.69
LMNA P02545 2/20 0.59
MEN1 O00255 2/20 0.59
KMT2A Q03164 2/20 0.59
TDP1 Q9NUW8 1/20 0.59
PGR P06401 2/20 0.58
AR P10275 2/20 0.58
CHRM1 P11229 1/20 0.58
CYP2C9 P11712 2/20 0.54
ABCB11 O95342 1/20 0.54
NR3C1 P04150 1/20 0.54
POLB P06746 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
HIF1A Q16665 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
CYP3A4 P08684 1/20 0.54
MAPK1 P28482 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6699256 0.82 CYP19A1 (1.00) CYP19A1PGRARCHRM1
SCHEMBL7592337 0.79 CYP19A1 (0.70) CYP19A1LMNAMEN1KMT2ATDP1
SCHEMBL144436 0.78 LMNA (0.72) CYP19A1LMNAMEN1KMT2ATDP1
SCHEMBL1650395 0.78 LMNA (0.72) CYP19A1LMNAMEN1KMT2ATDP1
SCHEMBL8859777 0.78 LMNA (0.67) CYP19A1LMNAMEN1KMT2ATDP1
SCHEMBL10868391 0.78 LMNA (0.72) CYP19A1LMNAMEN1KMT2ATDP1
SCHEMBL10444545 0.77 LMNA (0.63) CYP19A1LMNAMEN1KMT2ATDP1
SCHEMBL369752 0.76 CYP3A4 (0.66) CYP19A1LMNAMEN1KMT2ATDP1
SCHEMBL6577137 0.76 PGR (0.69) CYP19A1LMNAMEN1KMT2ATDP1
SCHEMBL18402585 0.76 CYP3A4 (0.66) CYP19A1LMNAMEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4416821-A Process for preparing 16-methylene steroids THE UPJOHN COMPANY (US) 1983-11-22 US claimed
EP-0402963-A2 17-Alpha ethynyl steroids THE UPJOHN COMPANY (US) 1990-12-19 EP disclosed
US-4614621-A Ethynylation of 16-methylene-17-keto steroids THE UPJOHN COMPANY (US) 1986-09-30 US disclosed
EP-0179496-A1 16-Sulfinylmethyl-steroids, their preparation and use THE UPJOHN COMPANY (US) 1986-04-30 EP disclosed
US-4567001-A 16-Methylene-17α-hydroxy-progesterones THE UPJOHN COMPANY (US) 1986-01-28 US disclosed
EP-0148616-A2 Stabilised monolithium acetylide and the ethynylation of steroids THE UPJOHN COMPANY (US) 1985-07-17 EP disclosed
US-4526720-A Process to prepare stabilized monolithium acetylide THE UPJOHN COMPANY (US) 1985-07-02 US disclosed
EP-0104054-A2 16-methylene-steroids and their preparation THE UPJOHN COMPANY (US) 1984-03-28 EP disclosed